SCHEMBL1729633

SCHEMBL1729633

Cc1cc(C(NC(=O)O)C2CCNCC2)nc(N)n1

nearest known ligand 0.42

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SMYD3 Q9H7B4 8/20 0.42
AKT1 P31749 9/20 0.38
CDK2 P24941 1/20 0.38
HRH4 Q9H3N8 1/20 0.37
GAA P10253 1/20 0.35
ATM Q13315 1/20 0.35
DNMT1 P26358 1/20 0.33
DNMT3L Q9UJW3 1/20 0.33
DNMT3A Q9Y6K1 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1727688 0.77 SMYD3 (0.43) SMYD3AKT1CDK2
SCHEMBL1727781 0.76 SMYD3 (0.43) SMYD3AKT1CDK2
SCHEMBL1728827 0.75 SMYD3 (0.44) SMYD3AKT1CDK2
SCHEMBL1729837 0.73 SMYD3 (0.42) SMYD3AKT1CDK2
SCHEMBL27600626 0.70 AKT1 (0.41) SMYD3AKT1CDK2
SCHEMBL1728854 0.70 AKT1 (0.45) SMYD3AKT1CDK2
SCHEMBL28037799 0.69 SMYD3 (0.46) SMYD3AKT1CDK2
SCHEMBL3701313 0.69 AKT1 (0.43) SMYD3AKT1CDK2
SCHEMBL4071612 0.68 SMYD3 (0.60) SMYD3AKT1CDK2
SCHEMBL1730307 0.68 KDM4E (0.46)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1633735-B1 DERIVATIVES OF PIPERIDINYL- AND PIPERAZINYL-ALKYL CARBAMATES, PREPARATION METHODS THEREOF AND APPLICATION OF SAME IN THERAPEUTICS SANOFI SA (FR) 2011-11-30 EP claimed