SCHEMBL3701313

SCHEMBL3701313

O=C(O)NC(c1ccncn1)C1CCNCC1

nearest known ligand 0.43

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 14/20 0.43
CDK2 P24941 1/20 0.43
SMYD3 Q9H7B4 6/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6066440 0.82 AAK1 (0.44) AKT1CDK2SMYD3
SCHEMBL27600626 0.80 AKT1 (0.41) AKT1CDK2SMYD3
SCHEMBL1729045 0.77 F11 (0.45) AKT1CDK2SMYD3
SCHEMBL1728006 0.75 P4HTM (0.37) AKT1CDK2SMYD3
SCHEMBL1728827 0.75 SMYD3 (0.44) AKT1CDK2SMYD3
SCHEMBL27655008 0.74 SLC6A4 (0.35) AKT1CDK2
SCHEMBL4071612 0.73 SMYD3 (0.60) AKT1CDK2SMYD3
SCHEMBL1727781 0.73 SMYD3 (0.43) AKT1CDK2SMYD3
SCHEMBL673132 0.71 CYP19A1 (0.37) AKT1
SCHEMBL30749440 0.71 CYP19A1 (0.37) AKT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2201012-A1 PYRROLO [2, 3 -D] PYRIMIDIN DERIVATIVES AS PROTEIN KINASE B INHIBITORS AstraZeneca AB (SE) 2010-06-30 EP disclosed
WO-2009047563-A1 PYRROLO [2, 3 -D] PYRIMIDIN DERIVATIVES AS PROTEIN KINASE B INHIBITORS ASTRAZENECA AB (SE) 2009-04-16 WO disclosed