SCHEMBL172981

SCHEMBL172981

CCc1cccc(-c2cccc(C(N)=O)c2)c1

nearest known ligand 0.61

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
BCL2 P10415 1/20 0.61
PTGS2 P35354 1/20 0.51
PARP1 P09874 6/20 0.50
AOC3 Q16853 2/20 0.49
ERN1 O75460 1/20 0.49
IDO1 P14902 1/20 0.47
DHODH Q02127 2/20 0.46
CSF1R P07333 1/20 0.46
FLT1 P17948 1/20 0.46
FLT3 P36888 1/20 0.46
CFD P00746 1/20 0.46
DHFR P00374 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL45866 0.89 PARP1 (0.57) BCL2PARP1
SCHEMBL10243328 0.88 BCL2 (0.55) BCL2PARP1AOC3ERN1DHODH
SCHEMBL10243641 0.88 BCL2 (0.55) BCL2PARP1AOC3ERN1DHODH
Hydrochloric Acid SCHEMBL27603084 0.87 PARP1 (0.55) BCL2PARP1
SCHEMBL12894987 0.84 BCL2 (0.78) BCL2PTGS2DHFR
SCHEMBL172996 0.84 CFD (0.61) PARP1AOC3ERN1DHODHCFD
SCHEMBL4940681 0.84 IKBKB (0.56) PARP1AOC3ERN1DHODHCFD
SCHEMBL31422694 0.83 PARP1 (0.64) PARP1ERN1DHODH
SCHEMBL2431097 0.83 PARP1 (0.64) PARP1ERN1DHODH
SCHEMBL12269244 0.83 ERN1 (0.49) PARP1AOC3ERN1DHODHCFD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019154366-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR AND USE THEREOF 江苏奥赛康药业有限公司 2019-08-15 WO disclosed
EP-1768966-B1 COUMPOUNDS AND METHODS FOR INHIBITING THE INTERACTION OF BCL PROTEINS WITH BINDING PARTNERS INFINITY DISCOVERY INC (US) 2012-03-07 EP disclosed