SCHEMBL17320249

SCHEMBL17320249

Cc1cc(Nc2nc(C3C4C=CC(C4)C3C(N)=O)c3ccccc3n2)ccc1OCCN1CCCC1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IRAK4 Q9NWZ3 8/20 0.58
MAP3K7 O43318 3/20 0.58
BACE1 P56817 2/20 0.42
AXL P30530 3/20 0.42
INSR P06213 2/20 0.42
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
SRC P12931 5/20 0.40
KDR P35968 3/20 0.40
YES1 P07947 1/20 0.40
EPHB4 P54760 1/20 0.40
BRD4 O60885 1/20 0.39
JAK1 P23458 1/20 0.39
HDAC1 Q13547 1/20 0.39
PDGFRB P09619 2/20 0.39
CDC7 O00311 1/20 0.39
PLK4 O00444 1/20 0.39
CHEK1 O14757 1/20 0.39
AURKA O14965 1/20 0.39
DCLK1 O15075 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1305489 0.87 IRAK4 (0.72) IRAK4MAP3K7AXLINSRSRC
SCHEMBL352214 0.79 IRAK4 (0.62) IRAK4MAP3K7BACE1INSRKDR
SCHEMBL30150294 0.74 IRAK4 (1.00) IRAK4MAP3K7AXLINSRSRC
SCHEMBL19742917 0.74 IRAK4 (1.00) IRAK4MAP3K7AXLINSRSRC
SCHEMBL14511547 0.73 MAP3K7 (0.44) IRAK4MAP3K7BACE1AXLINSR
SCHEMBL352672 0.70 IRAK4 (0.62) IRAK4MAP3K7AXLINSRSRC
SCHEMBL14483998 0.70 IRAK4 (0.62) IRAK4MAP3K7AXLINSRSRC
SCHEMBL349754 0.69 IRAK4 (0.80) IRAK4MAP3K7AXLINSRSRC
SCHEMBL10171322 0.68 IRAK4 (0.60) IRAK4MAP3K7INSRKDRMET
SCHEMBL10171268 0.68 IRAK4 (0.60) IRAK4MAP3K7AXLINSRSRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1960372-B1 KINASE INHIBITORS AND THEIR USES RIGEL PHARMACEUTICALS INC (US) 2015-12-09 EP disclosed