SCHEMBL17325533

SCHEMBL17325533

Cc1c(Cl)cccc1-c1cc(NC(C)c2ccccc2)nc(N)n1

nearest known ligand 0.56

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NUDT1 P36639 5/20 0.56
PFKFB3 Q16875 6/20 0.44
LDHA P00338 3/20 0.43
LDHB P07195 3/20 0.43
MAPK14 Q16539 1/20 0.43
HSP90AA1 P07900 1/20 0.43
HSP90AB1 P08238 1/20 0.43
TPH1 P17752 1/20 0.41
AGPAT2 O15120 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22839471 1.00 NUDT1 (0.56) NUDT1PFKFB3LDHALDHBMAPK14
SCHEMBL15757433 1.00 NUDT1 (0.56) NUDT1PFKFB3LDHALDHBMAPK14
SCHEMBL15756909 0.87 NUDT1 (0.56) NUDT1MAPK14HSP90AA1HSP90AB1AGPAT2
SCHEMBL28043729 0.85 NUDT1 (0.53) NUDT1PFKFB3LDHALDHBMAPK14
SCHEMBL28043730 0.85 NUDT1 (0.53) NUDT1PFKFB3LDHALDHBMAPK14
SCHEMBL15757415 0.80 NUDT1 (0.77) NUDT1HSP90AA1HSP90AB1AGPAT2
SCHEMBL17315318 0.79 HRH4 (0.55) NUDT1MAPK14HSP90AA1HSP90AB1AGPAT2
SCHEMBL20878223 0.78 NUDT1 (0.88) NUDT1TPH1
SCHEMBL17560838 0.78 NUDT1 (0.88) NUDT1TPH1
SCHEMBL17560919 0.77 NUDT1 (0.71) NUDT1HSP90AA1HSP90AB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106794181-A MTH1 inhibitors for the treatment of inflammatory and autoimmune conditions 托马斯·黑勒戴药物研究基金会 2017-05-31 CN disclosed
WO-2015187089-A1 MTH1 INHIBITORS FOR TREATMENT OF INFLAMMATORY AND AUTOIMMUNE CONDITIONS THOMAS HELLEDAYS STIFTELSE FÖR MEDICINSK FORSKNING (SE) 2015-12-10 WO disclosed