SCHEMBL28043729

SCHEMBL28043729

C[C@@H](Nc1cc(-c2cccc(Cl)c2CN)nc(N)n1)c1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NUDT1 P36639 4/20 0.53
TPH1 P17752 1/20 0.41
MAPK14 Q16539 1/20 0.41
HSP90AA1 P07900 1/20 0.40
HSP90AB1 P08238 1/20 0.40
PFKFB3 Q16875 4/20 0.40
AGPAT2 O15120 1/20 0.39
LDHA P00338 1/20 0.38
LDHB P07195 1/20 0.38
HRH4 Q9H3N8 4/20 0.38
HTR7 P34969 2/20 0.36
MAP4K4 O95819 1/20 0.36
ADRA1D P25100 1/20 0.36
ADRA1A P35348 1/20 0.36
ADRA1B P35368 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28043730 1.00 NUDT1 (0.53) NUDT1TPH1MAPK14HSP90AA1HSP90AB1
SCHEMBL28267202 0.88 NUDT1 (0.53) NUDT1MAPK14HSP90AA1HSP90AB1AGPAT2
SCHEMBL17325533 0.85 NUDT1 (0.56) NUDT1TPH1MAPK14HSP90AA1HSP90AB1
SCHEMBL22839471 0.85 NUDT1 (0.56) NUDT1TPH1MAPK14HSP90AA1HSP90AB1
SCHEMBL15757433 0.85 NUDT1 (0.56) NUDT1TPH1MAPK14HSP90AA1HSP90AB1
SCHEMBL28043809 0.81 NUDT1 (0.71) NUDT1HSP90AA1HSP90AB1AGPAT2HRH4
SCHEMBL28043763 0.79 NUDT1 (0.54) NUDT1HSP90AA1HSP90AB1AGPAT2HRH4
SCHEMBL28267599 0.78 NUDT1 (0.48) NUDT1MAPK14HSP90AA1HSP90AB1AGPAT2
SCHEMBL20878223 0.75 NUDT1 (0.88) NUDT1TPH1HRH4HTR7MAP4K4
SCHEMBL17560838 0.75 NUDT1 (0.88) NUDT1TPH1HRH4HTR7MAP4K4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105143206-B Pyrimidine -2,4- diamine derivative for treating cancer 托马斯·黑勒戴药物研究基金会 2019-01-15 CN claimed
CN-105143206-B Pyrimidine -2,4- diamine derivative for treating cancer 托马斯·黑勒戴药物研究基金会 2019-01-15 CN disclosed
CN-105143206-A Pyrimidine-2,4-diamine derivatives for treatment of cancer THOMAS HELLEDAYS STIFTELSE F R MEDICINSK FORSKNING 2015-12-09 CN disclosed