SCHEMBL17327809

SCHEMBL17327809

CC(=O)C1(c2ccccc2)Cc2ccccc2C1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC9 Q9UKV0 1/20 0.62
AKR1C1 Q04828 1/20 0.47
HDAC4 P56524 3/20 0.43
OPRM1 P35372 3/20 0.41
OPRD1 P41143 2/20 0.41
HSD11B1 P28845 2/20 0.41
OPRL1 P41146 1/20 0.41
ALOX15 P16050 1/20 0.41
SLC22A1 O15245 1/20 0.41
SLC6A4 P31645 1/20 0.41
ADRA1A P35348 1/20 0.41
OPRK1 P41145 1/20 0.41
KCNH2 Q12809 1/20 0.41
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA7 P43166 1/20 0.40
CA9 Q16790 1/20 0.40
CA14 Q9ULX7 1/20 0.40
P2RX7 Q99572 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15215650 0.86 AKR1C1 (0.48) HDAC9AKR1C1HDAC4OPRM1OPRD1
SCHEMBL10571417 0.83 HDAC9 (0.67) HDAC9AKR1C1HDAC4HSD11B1ALOX15
SCHEMBL890180 0.81 AKR1C1 (0.57) HDAC9AKR1C1HDAC4OPRM1OPRD1
SCHEMBL3737199 0.78 AKR1C1 (0.70) AKR1C1HDAC4OPRD1HSD11B1CA12
SCHEMBL12928712 0.78 AKR1C1 (0.64) AKR1C1HDAC4OPRD1HSD11B1CA12
SCHEMBL17316173 0.77 HDAC9 (1.00) HDAC9AKR1C1HDAC4
SCHEMBL24663621 0.76 AKR1C1 (0.52) HDAC9AKR1C1HDAC4OPRM1OPRD1
SCHEMBL1838291 0.76 AKR1C1 (0.68) AKR1C1HDAC4HSD11B1P2RX7
SCHEMBL8324812 0.76 OPRM1 (0.63) OPRM1OPRD1HSD11B1SLC22A1SLC6A4
SCHEMBL17316010 0.75 OPRM1 (0.67) HDAC9OPRM1OPRD1SLC22A1SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015187542-A1 HISTONE DEACETYLASE INHIBITORS AND COMPOSITIONS AND METHODS OF USE THEREOF CHDI FOUNDATION INC. (US) 2015-12-10 WO disclosed