SCHEMBL17336302

SCHEMBL17336302

O=c1[nH]c(-c2cc[nH]n2)nc2ccccc12

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.61
NPC1 O15118 2/20 0.61
RAB9A P51151 2/20 0.61
LMNA P02545 1/20 0.61
GAA P10253 1/20 0.61
HTT P42858 1/20 0.61
HIF1A Q16665 1/20 0.61
L3MBTL1 Q9Y468 1/20 0.61
TNKS O95271 8/20 0.61
TNKS2 Q9H2K2 8/20 0.61
PARP1 P09874 5/20 0.61
HPGD P15428 4/20 0.55
MAPT P10636 1/20 0.55
ALOX15 P16050 1/20 0.55
HSD17B10 Q99714 1/20 0.55
APOBEC3G Q9HC16 1/20 0.55
GUSB P08236 7/20 0.54
PARP2 Q9UGN5 2/20 0.54
KDM4E B2RXH2 2/20 0.54
CYP1A1 P04798 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6695759 0.81 TNKS2 (0.81) ALDH1A1NPC1RAB9ALMNAGAA
SCHEMBL12758425 0.80 ALDH1A1 (0.73) ALDH1A1NPC1RAB9ALMNAGAA
SCHEMBL29941412 0.77 NPC1 (0.62) ALDH1A1NPC1RAB9ALMNAGAA
SCHEMBL546102 0.77 NPC1 (0.62) ALDH1A1NPC1RAB9ALMNAGAA
SCHEMBL6885282 0.76 TNKS (0.93) ALDH1A1NPC1RAB9ATNKSTNKS2
SCHEMBL258433 0.76 TNKS (1.00) ALDH1A1NPC1RAB9ATNKSTNKS2
SCHEMBL29592833 0.76 TNKS (1.00) ALDH1A1NPC1RAB9ATNKSTNKS2
SCHEMBL29764050 0.76 NPC1 (1.00) ALDH1A1NPC1RAB9ALMNAGAA
SCHEMBL10709261 0.76 NPC1 (1.00) ALDH1A1NPC1RAB9ALMNAGAA
SCHEMBL21843249 0.76 ALDH1A1 (0.63) ALDH1A1NPC1RAB9ALMNAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114621194-B 4-methylene-N-hydroxybenzoamide compound and application thereof 沈阳药科大学 2023-08-29 CN disclosed
CN-114621194-B 4-methylene-N-hydroxybenzoamide compound and application thereof 沈阳药科大学 2023-08-29 CN disclosed
CN-114621194-A 4-methylene-N-hydroxybenzamide compound and application thereof 沈阳药科大学 2022-06-14 CN disclosed
EP-3154961-A1 QUINAZOLINONE DERIVATIVES AS PHOSPHATIDYLINOSITOL 3-KINASE INHIBITORS Gilead Sciences, Inc. (US) 2017-04-19 EP disclosed
WO-2015191743-A1 QUINAZOLINONE DERIVATIVES AS PHOSPHATIDYLINOSITOL 3-KINASE INHIBITORS GILEAD SCIENCES, INC. (US) 2015-12-17 WO disclosed