SCHEMBL258433

SCHEMBL258433

O=c1[nH]c(-c2ccccc2)nc2ccccc12

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TNKS O95271 13/20 1.00
TNKS2 Q9H2K2 12/20 1.00
PARP1 P09874 6/20 1.00
HPGD P15428 2/20 0.81
MAPT P10636 2/20 0.81
ALDH1A1 P00352 1/20 0.81
ALOX15 P16050 1/20 0.81
HSD17B10 Q99714 1/20 0.81
APOBEC3G Q9HC16 1/20 0.81
GUSB P08236 6/20 0.78
PARP2 Q9UGN5 3/20 0.78
CYP1A1 P04798 1/20 0.78
CYP1B1 Q16678 1/20 0.78
NPC1 O15118 3/20 0.71
RAB9A P51151 3/20 0.71
WNT3A P56704 1/20 0.71
CASP3 P42574 1/20 0.71
SENP7 Q9BQF6 1/20 0.71
SENP6 Q9GZR1 1/20 0.71
KDM4E B2RXH2 1/20 0.71

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29592833 1.00 TNKS (1.00) TNKSTNKS2PARP1HPGDMAPT
Hydrochloric Acid SCHEMBL31529601 0.98 TNKS (0.96) TNKSTNKS2PARP1HPGDMAPT
SCHEMBL6124189 0.96 TNKS (0.93) TNKSTNKS2PARP1HPGDMAPT
SCHEMBL6885282 0.96 TNKS (0.93) TNKSTNKS2PARP1HPGDMAPT
SCHEMBL8620410 0.91 TNKS (0.83) TNKSTNKS2PARP1HPGDMAPT
SCHEMBL6695759 0.90 TNKS2 (0.81) TNKSTNKS2PARP1HPGDMAPT
SCHEMBL29831923 0.90 HPGD (1.00) TNKSTNKS2PARP1HPGDMAPT
SCHEMBL3460177 0.90 HPGD (1.00) TNKSTNKS2PARP1HPGDMAPT
SCHEMBL16768506 0.88 TNKS (0.78) TNKSTNKS2PARP1HPGDMAPT
SCHEMBL8618982 0.88 TNKS (1.00) TNKSTNKS2PARP1HPGDMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 279 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118027093-A Siloxane ligand protected V6Nanocluster, synthesis method and catalytic application thereof 山东交通学院 2024-05-14 CN claimed
EP-4008716-A1 NOVEL INHIBITORS OF INSULIN-LIKE GROWTH FACTOR 2 MRNA BINDING PROTEINS Martin-Luther-Universität Halle-Wittenberg (DE) 2022-06-08 EP claimed
EP-4008717-A2 NOVEL INHIBITORS OF INSULIN-LIKE GROWTH FACTOR 2 MRNA BINDING PROTEINS Martin-Luther-Universität Halle-Wittenberg (DE) 2022-06-08 EP claimed
EP-3160960-A1 PHOSPHATIDYLINOSITOL 3-KINASE INHIBITORS GILEAD SCIENCES, INC. (US) 2017-05-03 EP claimed
WO-2015200352-A1 PHOSPHATIDYLINOSITOL 3-KINASE INHIBITORS GILEAD SCIENCES, INC. (US) 2015-12-30 WO claimed
EP-1761540-A1 QUINAZOLINONES AS INHIBITORS OF HUMAN PHOSPHATIDYLINOSITOL 3-KINASE DELTA ICOS CORPORATION (US) 2007-03-14 EP claimed
WO-2005113556-A1 QUINAZOLINONES AS INHIBITORS OF HUMAN PHOSPHATIDYLINOSITOL 3-KINASE DELTA ICOS CORPORATION (US) 2005-12-01 WO claimed
US-6479499-B1 INHIBITORS OF TUBULIN POLYMERIZATION NATIONAL SCIENCE COUNCIL (TW) 2002-11-12 US claimed
CN-115650924-B Green synthesis method of quinazolinone 山东华泰新材料技术研发有限公司 2024-08-20 CN disclosed
CN-118027093-A Siloxane ligand protected V6Nanocluster, synthesis method and catalytic application thereof 山东交通学院 2024-05-14 CN disclosed
CN-117964560-A Method for constructing quinazolinone derivative through oxidization 淮阴工学院 2024-05-03 CN disclosed
CN-117561063-A Heterocyclic compounds and methods of use 安进公司 2024-02-13 CN disclosed
CN-111777564-B Method for synthesizing quinazolinone compound by photocatalytic alcohol oxidation in aqueous phase 许昌学院 2023-07-14 CN disclosed
CN-114591251-B Chiral aminoquinazoline compound, and preparation method and application thereof 华南理工大学 2023-06-20 CN disclosed
EP-0013612-A2 (Piperidinylalkyl)quinazoline derivatives, process for their preparation and pharmaceutical compositions containing them JANSSEN PHARMACEUTICA N.V. (BE) 1980-07-23 EP disclosed
US-4159330-A ANTIALLERGENS CARLO ERBA S.P.A. (IT) 1979-06-26 US disclosed
US-4159330-A ANTIALLERGENS CARLO ERBA S.P.A. (IT) 1979-06-26 US disclosed
US-3998951-A Substituted 2-arylquinazolines as fungicides FMC CORPORATION (US) 1976-12-21 US disclosed
US-3932409-A CYTOSTATIC AGENTS BAYER AKTIENGESELLSCHAFT (DT) 1976-01-13 US disclosed
US-3932409-A CYTOSTATIC AGENTS BAYER AKTIENGESELLSCHAFT (DT) 1976-01-13 US disclosed