SCHEMBL17339124

SCHEMBL17339124

CCOC(=O)c1ccc2ccccn12

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.51
ALDH1A1 P00352 6/20 0.50
KDM4E B2RXH2 4/20 0.50
GAA P10253 4/20 0.50
HPGD P15428 2/20 0.50
GLA P06280 1/20 0.50
HTT P42858 1/20 0.50
ATM Q13315 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
TSHR P16473 2/20 0.49
CYP1A2 P05177 6/20 0.47
CYP2C9 P11712 4/20 0.47
CYP2C19 P33261 4/20 0.47
SMN1; SMN2 Q16637 3/20 0.47
NPSR1 Q6W5P4 1/20 0.47
RXFP1 Q9HBX9 1/20 0.47
CYP3A4 P08684 4/20 0.45
PTGS1 P23219 1/20 0.45
PTGS2 P35354 1/20 0.45
IDO1 P14902 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27984769 0.89 SMN1; SMN2 (0.48) MAPK1ALDH1A1KDM4EGAAHPGD
SCHEMBL6219618 0.86 MAPK1 (0.48) MAPK1ALDH1A1KDM4EGAAHPGD
SCHEMBL25515640 0.81 MAPT (0.48) MAPK1ALDH1A1KDM4EGAAHPGD
SCHEMBL8122403 0.81 HTT (0.45) MAPK1ALDH1A1KDM4EGAAHPGD
SCHEMBL4616746 0.80 KDM4E (0.64) MAPK1ALDH1A1KDM4EGAAHPGD
SCHEMBL6248007 0.78 L3MBTL1 (0.40) MAPK1ALDH1A1KDM4EGAAHPGD
SCHEMBL21358704 0.77 MEN1 (0.41) HTTATML3MBTL1MEN1KMT2A
SCHEMBL14963083 0.76 KDM4E (0.49) MAPK1ALDH1A1KDM4EGAAHPGD
SCHEMBL14963077 0.75 ALDH1A1 (0.48) MAPK1ALDH1A1KDM4EGAAHPGD
SCHEMBL17339205 0.75 KDM4E (0.58) MAPK1ALDH1A1KDM4EGAAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111892579-B Kinase inhibitors 上海艾力斯医药科技股份有限公司 2023-07-25 CN disclosed
CN-116134035-A 3- (1H-imidazol-2-yl) -2,3,8 a-tetrahydroindol-5 (1H) -one derivatives useful as factor XIA inhibitors 詹森药业有限公司 2023-05-16 CN disclosed
CN-111892579-A Kinase inhibitor 上海复尚慧创医药研究有限公司 2020-11-06 CN disclosed
CN-111875585-A Kinase inhibitor 上海复尚慧创医药研究有限公司 2020-11-03 CN disclosed
CN-106660993-B Kinase inhibitor 上海复尚慧创医药研究有限公司 2020-09-11 CN disclosed
CN-106660993-A Kinase inhibitor 上海复尚慧创医药研究有限公司 2017-05-10 CN disclosed
WO-2015188777-A1 CERTAIN PROTEIN KINASE INHIBITORS SHANGHAI FOCHON PHARMACEUTICAL CO LTD (CN) 2015-12-17 WO disclosed