SCHEMBL17339656

SCHEMBL17339656

C=C(C(N)=O)c1ccc(OC)nc1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NNMT P40261 5/20 0.70
MKNK1 Q9BUB5 1/20 0.58
MKNK2 Q9HBH9 1/20 0.58
SIRT6 Q8N6T7 1/20 0.45
MAPT P10636 2/20 0.42
MAOA P21397 1/20 0.42
MAOB P27338 1/20 0.42
OXTR P30559 1/20 0.42
KLK3 P07288 1/20 0.41
KDM4E B2RXH2 2/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
RAB9A P51151 3/20 0.40
NPC1 O15118 2/20 0.40
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.40
HTT P42858 1/20 0.40
GPR183 P32249 3/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
PABPC1 P11940 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30475723 1.00 NNMT (0.70) NNMTMKNK1MKNK2SIRT6MAPT
SCHEMBL30475743 0.85 NNMT (0.62) NNMTMKNK1MKNK2MAPTMAOA
SCHEMBL8664420 0.83 NNMT (0.60) NNMTMKNK1MKNK2MAPTMAOA
SCHEMBL28522209 0.83 NNMT (0.49) NNMTMKNK1MKNK2MAPT
SCHEMBL29975550 0.82 NNMT (1.00) NNMTMKNK1MKNK2SIRT6MAPT
SCHEMBL71905 0.82 NNMT (1.00) NNMTMKNK1MKNK2SIRT6MAPT
SCHEMBL1515510 0.81 NNMT (0.72) NNMTMKNK1MKNK2SIRT6MAPT
Hydrochloric Acid SCHEMBL5013391 0.81 NNMT (0.96) NNMTMKNK1MKNK2SIRT6MAPT
Hydrochloric Acid SCHEMBL6234386 0.81 NNMT (0.96) NNMTMKNK1MKNK2SIRT6MAPT
SCHEMBL18228074 0.78 NNMT (0.72) NNMTMKNK1MKNK2SIRT6MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111875585-B Kinase inhibitors 上海艾力斯医药科技股份有限公司 2023-06-23 CN disclosed
CN-112409360-B Heteroaryl vinyl xanthine derivatives and uses thereof 广东东阳光药业有限公司 2022-12-23 CN disclosed
CN-112409360-A Heteroaryl vinyl xanthine derivatives and uses thereof 广东东阳光药业有限公司 2021-02-26 CN disclosed
CN-111892579-A Kinase inhibitor 上海复尚慧创医药研究有限公司 2020-11-06 CN disclosed
CN-111875585-A Kinase inhibitor 上海复尚慧创医药研究有限公司 2020-11-03 CN disclosed
CN-106660993-B Kinase inhibitor 上海复尚慧创医药研究有限公司 2020-09-11 CN disclosed
WO-2015188777-A1 CERTAIN PROTEIN KINASE INHIBITORS SHANGHAI FOCHON PHARMACEUTICAL CO LTD (CN) 2015-12-17 WO disclosed