SCHEMBL17354485

SCHEMBL17354485

NCCCN(CCCN)Cc1ccc(-c2c[nH]c(NC(=O)Nc3ccccc3OCF)nc2=O)cc1

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
IGF1R P08069 4/20 0.36
P2RY1 P47900 1/20 0.33
HDAC1 Q13547 1/20 0.33
ROCK2 O75116 1/20 0.32
LIMK1 P53667 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
KMT2A Q03164 3/20 0.32
MEN1 O00255 1/20 0.32
GAA P10253 1/20 0.32
MAPT P10636 2/20 0.31
IMPDH2 P12268 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
LMNA P02545 1/20 0.30
TP53 P04637 1/20 0.30
POLB P06746 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17486576 0.94 IGF1R (0.35) IGF1RP2RY1HDAC1KMT2AMEN1
SCHEMBL17486581 0.94 IGF1R (0.33) IGF1RP2RY1
SCHEMBL17486543 0.93 KMT2A (0.34) IGF1RP2RY1HDAC1KMT2AMEN1
SCHEMBL17486575 0.93 IGF1R (0.33) IGF1RP2RY1
SCHEMBL17486553 0.92 IGF1R (0.33) IGF1RP2RY1ROCK2LIMK1
SCHEMBL17486568 0.92 HDAC1 (0.36) IGF1RP2RY1HDAC1KMT2AMEN1
SCHEMBL13589 0.90 KDR (0.40) IGF1RP2RY1HDAC1
SCHEMBL17486554 0.89 P2RY1 (0.35) IGF1RP2RY1MAPT
SCHEMBL13975 0.88 KDR (0.38) IGF1RP2RY1HDAC1
SCHEMBL13963 0.87 KDR (0.38) IGF1RP2RY1HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9216979-B2 Antimicrobial compounds and methods of making and using the same MELINTA THERAPEUTICS, INC. (US) 2015-12-22 US disclosed