SCHEMBL1735518

SCHEMBL1735518

CC(Cc1ccccc1)Nc1nc(C(N)=O)cc(-c2ccccc2)n1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.50
FPR2 P25090 1/20 0.49
SCN9A Q15858 1/20 0.49
ADORA1 P30542 7/20 0.46
GLA P06280 2/20 0.45
HTT P42858 2/20 0.45
ALDH1A1 P00352 3/20 0.44
HPGD P15428 2/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
HSD17B10 Q99714 3/20 0.44
GAA P10253 1/20 0.44
TSHR P16473 1/20 0.44
CASP1 P29466 1/20 0.44
CASP7 P55210 1/20 0.44
ADORA3 P0DMS8 2/20 0.43
ADORA2A P29274 1/20 0.43
ADORA2B P29275 1/20 0.43
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1733575 0.85 FPR2 (0.55) KDM4EFPR2SCN9AADORA1GLA
SCHEMBL1734509 0.84 KDM4E (0.49) KDM4EFPR2SCN9AADORA1GLA
SCHEMBL1734121 0.84 KDM4E (0.51) KDM4EFPR2SCN9AADORA1GLA
SCHEMBL1735520 0.81 KDM4E (0.56) KDM4EFPR2SCN9AADORA1GLA
SCHEMBL1734267 0.80 PIK3CB (0.57) KDM4EGLAHTTALDH1A1HPGD
SCHEMBL1735244 0.80 FPR2 (0.50) KDM4EFPR2SCN9AADORA1GLA
SCHEMBL1734424 0.79 KDM4E (0.53) KDM4EFPR2SCN9AADORA1GLA
SCHEMBL3718054 0.78 GRM2 (0.46) KDM4EFPR2SCN9AMEN1KMT2A
SCHEMBL1733664 0.78 TDP1 (0.65) KDM4EFPR2SCN9AADORA1GLA
SCHEMBL3721016 0.78 SCN9A (0.48) FPR2SCN9AMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1891018-B1 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS VERTEX PHARMA (US) 2011-11-16 EP claimed
WO-2011131686-A1 A THERMALLY CONTROLLED ASSEMBLY NAPATECH A/S (DK) 2011-10-27 WO claimed