SCHEMBL1735520

SCHEMBL1735520

CCC(CC)Nc1nc(C(N)=O)cc(-c2ccccc2)n1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.56
ADORA1 P30542 11/20 0.52
FPR2 P25090 1/20 0.49
SCN9A Q15858 1/20 0.49
ADORA3 P0DMS8 3/20 0.49
ADORA2A P29274 3/20 0.49
ADORA2B P29275 1/20 0.49
GLA P06280 2/20 0.47
HTT P42858 2/20 0.47
ALDH1A1 P00352 3/20 0.46
HPGD P15428 2/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
HSD17B10 Q99714 3/20 0.46
GAA P10253 1/20 0.46
TSHR P16473 1/20 0.46
CASP1 P29466 1/20 0.46
CASP7 P55210 1/20 0.46
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1734431 0.92 KDM4E (0.51) KDM4EADORA1FPR2SCN9AADORA3
SCHEMBL1734181 0.91 KDM4E (0.50) KDM4EADORA1FPR2SCN9AADORA3
SCHEMBL1734296 0.89 KDM4E (0.48) KDM4EADORA1FPR2SCN9AADORA3
SCHEMBL1733575 0.85 FPR2 (0.55) KDM4EADORA1FPR2SCN9AADORA3
SCHEMBL1734509 0.85 KDM4E (0.49) KDM4EADORA1FPR2SCN9AADORA3
SCHEMBL1734332 0.83 KDM4E (0.60) KDM4EADORA1ADORA3ADORA2AADORA2B
SCHEMBL1734121 0.82 KDM4E (0.51) KDM4EADORA1FPR2SCN9AADORA3
SCHEMBL1735518 0.81 KDM4E (0.50) KDM4EADORA1FPR2SCN9AADORA3
SCHEMBL1733664 0.81 TDP1 (0.65) KDM4EADORA1FPR2SCN9AADORA3
SCHEMBL1734127 0.81 KDM4E (0.57) KDM4EADORA1ADORA3ADORA2AADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1891018-B1 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS VERTEX PHARMA (US) 2011-11-16 EP claimed
WO-2011131686-A1 A THERMALLY CONTROLLED ASSEMBLY NAPATECH A/S (DK) 2011-10-27 WO claimed