SCHEMBL17366170

SCHEMBL17366170

O=C(c1ccccc1)c1ccc(CN2C(=O)c3ccccc3C2c2ccc(Cl)cc2)cc1

nearest known ligand 0.64

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MDM2 Q00987 7/20 0.64
TP53 P04637 3/20 0.55
ALDH1A1 P00352 2/20 0.48
GAA P10253 1/20 0.47
HTT P42858 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
ATM Q13315 1/20 0.47
MAPT P10636 1/20 0.44
PRKAG1 P54619 1/20 0.44
PRKAA2 P54646 1/20 0.44
PRKAB1 Q9Y478 1/20 0.44
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30121977 0.90 MDM2 (0.64) MDM2TP53ALDH1A1GAAHTT
SCHEMBL17366156 0.89 MDM2 (0.60) MDM2TP53ALDH1A1GAAHTT
SCHEMBL17366151 0.84 MDM2 (0.58) MDM2TP53ALDH1A1GAAHTT
SCHEMBL17366174 0.84 MDM2 (0.58) MDM2TP53ALDH1A1GAAHTT
SCHEMBL17366169 0.84 MDM2 (0.58) MDM2TP53ALDH1A1GAAHTT
SCHEMBL17366179 0.81 MDM2 (0.55) MDM2TP53ALDH1A1MAPTMEN1
SCHEMBL17366150 0.81 MDM2 (0.55) MDM2TP53ALDH1A1GAAHTT
SCHEMBL8274847 0.80 MEN1 (0.55) MDM2ALDH1A1GAAHTTNPSR1
SCHEMBL17366148 0.80 CYP2C9 (0.57) MDM2TP53MEN1KMT2A
SCHEMBL8272076 0.79 TP53 (0.59) MDM2TP53ALDH1A1GAAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2960233-B1 NEW THERAPEUTIC AGENTS CANCER RESEARCH TECH LTD (GB) 2019-10-30 EP disclosed
US-10414726-B2 Therapeutic agents CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2019-09-17 US disclosed
US-20180118684-A1 THERAPEUTIC AGENTS CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2018-05-03 US disclosed
EP-2960233-A1 NEW THERAPEUTIC AGENTS Cancer Research Technology Limited (GB) 2015-12-30 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180118684-A1 THERAPEUTIC AGENTS TP53, MDM2, TP53BP1 MDM2 2/4885TP53 1/4885ALDH1A1 2445/4885
US-10414726-B2 Therapeutic agents TP53, MDM2, TP53BP1 MDM2 2/4885TP53 1/4885ALDH1A1 2445/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.