SCHEMBL17366201

SCHEMBL17366201

O=Nc1ccc(CN2C(=O)c3ccc(F)c(Cl)c3C2c2ccc(Cl)cc2)cc1

nearest known ligand 0.50

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MDM2 Q00987 8/20 0.50
TP53 P04637 5/20 0.41
MAPT P10636 2/20 0.34
RXFP1 Q9HBX9 1/20 0.32
PTDSS1 P48651 1/20 0.32
TRPM8 Q7Z2W7 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17366184 0.82 MDM2 (0.46) MDM2TP53
SCHEMBL17366169 0.69 MDM2 (0.58) MDM2TP53MAPTTRPM8
SCHEMBL30121977 0.68 MDM2 (0.64) MDM2TP53MAPT
SCHEMBL17366161 0.66 MDM2 (0.51) MDM2TP53MAPT
SCHEMBL29872333 0.65 TP53 (0.38) MDM2TP53MAPTPTDSS1
SCHEMBL17366153 0.65 MDM2 (0.52) MDM2TP53
SCHEMBL17366182 0.65 MDM2 (0.56) MDM2TP53MAPT
SCHEMBL31520186 0.65 MDM2 (0.45) MDM2TP53MAPTRXFP1PTDSS1
SCHEMBL30122194 0.64 MDM2 (0.41) MDM2TP53
SCHEMBL17366151 0.64 MDM2 (0.58) MDM2TP53MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2960233-B1 NEW THERAPEUTIC AGENTS CANCER RESEARCH TECH LTD (GB) 2019-10-30 EP disclosed
EP-2960233-A1 NEW THERAPEUTIC AGENTS Cancer Research Technology Limited (GB) 2015-12-30 EP disclosed