SCHEMBL1736800

SCHEMBL1736800

C#CCn1c(C)c(C)c2ccnc(-c3ccc(OC)cc3)c21

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.51
MEN1 O00255 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
KMT2A Q03164 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
DYRK1A Q13627 5/20 0.38
MAOA P21397 1/20 0.38
PDE3B Q13370 1/20 0.38
PDE3A Q14432 1/20 0.38
KDM4E B2RXH2 3/20 0.37
ALDH1A1 P00352 3/20 0.37
HPGD P15428 1/20 0.37
CASR P41180 1/20 0.36
CCNA2 P20248 1/20 0.36
CDK2 P24941 1/20 0.36
PTGS2 P35354 1/20 0.36
DYRK3 O43781 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL1736348 0.99 ACHE (0.50) ACHEMEN1CYP3A4CYP2D6CYP2C9
SCHEMBL1737399 0.88 ACHE (0.39) ACHEMEN1CYP3A4CYP2C19KMT2A
Hydrochloric Acid SCHEMBL1737857 0.86 ACHE (0.38) ACHEMEN1CYP3A4CYP2C19KMT2A
SCHEMBL1736111 0.85 ACHE (0.37) ACHEMEN1KMT2ANPSR1PDE3B
SCHEMBL1738139 0.85 ACHE (0.37) ACHEMEN1CYP2C9CYP2C19KMT2A
SCHEMBL1738462 0.85 DYRK1A (0.47) CYP3A4CYP2D6CYP2C19DYRK1APDE3B
Hydrochloric Acid SCHEMBL1735787 0.84 ACHE (0.37) ACHEMEN1KMT2ANPSR1PDE3B
Hydrochloric Acid SCHEMBL1737854 0.84 ACHE (0.37) ACHENPSR1PDE3BPDE3AKDM4E
Hydrochloric Acid SCHEMBL1735573 0.84 DYRK1A (0.46) CYP3A4CYP2D6CYP2C19DYRK1APDE3B
SCHEMBL1739797 0.83 ALDH1A1 (0.46) MEN1CYP3A4KMT2ANPSR1PDE3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1784404-B1 PYRROLO[2,3-C]PYRIDINE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF YUHAN CORP (KR) 2011-11-16 EP claimed
US-20110263306-A1 COMPUTER SYSTEM AND PROGRAM NAMCO BANDAI GAMES INC. (JP) 2011-10-27 US claimed
EP-1784404-A4 PYRROLO[2,3-C]PYRIDINE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF YUHAN CORP (KR) 2009-09-09 EP claimed
JP-2008511621-A 2008-04-17 JP claimed
EP-1784404-A1 PYRROLO[2,3-C]PYRIDINE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF Yuhan Corporation (KR) 2007-05-16 EP claimed
WO-2006025716-A1 PYRROLO[2,3-C]PYRIDINE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF YUHAN CORPORATION (KR) 2006-03-09 WO claimed