SCHEMBL17375418

SCHEMBL17375418

O=C(O)c1cccc(Br)c1F.O=C(O)c1ccccc1F

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALB P02768 1/20 0.52
CES2 O00748 2/20 0.48
CES1 P23141 2/20 0.48
PRNP P04156 1/20 0.47
ALDH1A1 P00352 4/20 0.46
ALOX15 P16050 2/20 0.46
BCHE P06276 1/20 0.46
MAOB P27338 1/20 0.43
FABP4 P15090 1/20 0.43
PTPN1 P18031 1/20 0.42
ERCC5 P28715 1/20 0.42
FEN1 P39748 1/20 0.42
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA4 P22748 1/20 0.42
CA7 P43166 1/20 0.42
CA9 Q16790 1/20 0.42
GAA P10253 1/20 0.42
ACMSD Q8TDX5 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29570698 0.91 PRNP (0.50) ALBCES2CES1PRNPALDH1A1
SCHEMBL146386 0.91 PRNP (0.50) ALBCES2CES1PRNPALDH1A1
SCHEMBL97828 0.82 CES2 (0.68) ALBCES2CES1ALDH1A1ALOX15
SCHEMBL29362443 0.82 CES2 (0.68) ALBCES2CES1ALDH1A1ALOX15
SCHEMBL30968201 0.82 CES2 (0.68) ALBCES2CES1ALDH1A1ALOX15
Hydrochloric Acid SCHEMBL23201659 0.80 CES2 (0.65) ALBCES2CES1ALDH1A1ALOX15
SCHEMBL10357059 0.80 CES2 (0.65) ALBCES2CES1ALDH1A1ALOX15
SCHEMBL11451385 0.80 CES2 (0.65) ALBCES2CES1ALDH1A1ALOX15
Hydrochloric Acid SCHEMBL6592453 0.80 CES2 (0.65) ALBCES2CES1ALDH1A1ALOX15
SCHEMBL9015790 0.80 CES2 (0.65) ALBCES2CES1ALDH1A1ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3160967-A1 IMIDAZO[1,2-A]PYRAZIN-1YL-BENZAMIDE COMPOUNDS FOR TREATING SPINAL MUSCULAR ATROPHY F. Hoffmann-La Roche AG (CH) 2017-05-03 EP disclosed
WO-2015197503-A1 IMIDAZO[1,2-A]PYRAZIN-1YL-BENZAMIDE COMPOUNDS FOR TREATING SPINAL MUSCULAR ATROPHY F. HOFFMANN-LA ROCHE AG (CH) 2015-12-30 WO disclosed