SCHEMBL17377199

SCHEMBL17377199

Nc1c(S(=O)(=O)c2ccccc2)c2ncnc(Cl)c2n1-c1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.47
ALDH1A1 P00352 3/20 0.47
GAA P10253 3/20 0.47
KMT2A Q03164 2/20 0.47
HPGD P15428 2/20 0.47
LMNA P02545 1/20 0.47
GLA P06280 1/20 0.45
MAPT P10636 1/20 0.45
TP53 P04637 1/20 0.43
FFAR2 O15552 16/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17377302 0.83 FFAR2 (0.47) KDM4EALDH1A1GAAKMT2AHPGD
SCHEMBL17377197 0.80 KDM4E (0.51) KDM4EALDH1A1GAAKMT2AHPGD
SCHEMBL17377290 0.77 KDM4E (0.47) KDM4EALDH1A1GAAKMT2AHPGD
SCHEMBL19743040 0.75 FFAR2 (0.48) KDM4EALDH1A1GAAFFAR2
SCHEMBL17376395 0.71 FFAR2 (0.70) FFAR2
SCHEMBL17379138 0.69 KDM4E (0.48) KDM4EALDH1A1GAAKMT2AHPGD
SCHEMBL17377218 0.68 ALDH1A1 (0.47) KDM4EALDH1A1GAAKMT2AHPGD
SCHEMBL17377301 0.66 FFAR2 (0.50) KDM4EALDH1A1GAAFFAR2
SCHEMBL17377182 0.66 FFAR2 (0.48) KDM4EALDH1A1GAAKMT2AHPGD
SCHEMBL17377310 0.65 GAA (0.51) KDM4EALDH1A1GAAKMT2AHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3160955-A1 1,3-SUBSTITUTED 2-AMINOINDOLE DERIVATIVES AND ANALOGUES USEFUL IN THE TREATMENT OR PREVENTION OF DIABETES MELLITUS, OBESITY AND INFLAMMATORY BOWEL DISEASE Takeda Pharmaceutical Company Limited (JP) 2017-05-03 EP disclosed
WO-2015198046-A1 1,3-SUBSTITUTED 2-AMINOINDOLE DERIVATIVES AND ANALOGUES USEFUL IN THE TREATMENT OR PREVENTION OF DIABETES MELLITUS, OBESITY AND INFLAMMATORY BOWEL DISEASE TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2015-12-30 WO disclosed