SCHEMBL17382010

SCHEMBL17382010

Cc1cnn(CC(N)=O)c1C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 4/20 0.41
GRIA1 P42261 1/20 0.39
GRIA2 P42262 1/20 0.39
GRIA3 P42263 1/20 0.39
GRIA4 P48058 1/20 0.39
TSHR P16473 1/20 0.35
SMN1; SMN2 Q16637 3/20 0.34
MITF O75030 3/20 0.34
ALDH1A1 P00352 3/20 0.34
MAPT P10636 3/20 0.34
RAB9A P51151 3/20 0.34
S1PR4 O95977 2/20 0.34
S1PR1 P21453 2/20 0.34
NPC1 O15118 2/20 0.34
TGFBR1 P36897 2/20 0.34
GAA P10253 2/20 0.33
CYP3A4 P08684 1/20 0.33
KDM4E B2RXH2 1/20 0.33
HTT P42858 3/20 0.32
NOS1 P29475 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17382258 0.81 LMNA (0.40) LMNASMN1; SMN2MITFALDH1A1MAPT
SCHEMBL19321628 0.79 LMNA (0.38) LMNASMN1; SMN2MITFALDH1A1MAPT
SCHEMBL19236923 0.75 SMN1; SMN2 (0.36) LMNAGRIA1GRIA2GRIA3GRIA4
SCHEMBL12985515 0.75 SMN1; SMN2 (0.54) LMNATSHRSMN1; SMN2ALDH1A1MAPT
SCHEMBL31131810 0.75 LMNA (0.42) LMNATSHRSMN1; SMN2ALDH1A1MAPT
SCHEMBL26722179 0.73
SCHEMBL1803436 0.71 TSHR (0.38) LMNATSHRSMN1; SMN2MITFALDH1A1
SCHEMBL1360243 0.70
SCHEMBL29078400 0.69 GRIA1 (0.39) GRIA1GRIA2GRIA3GRIA4NOS1
SCHEMBL12121230 0.69 POLB (0.40) LMNAGRIA1GRIA2GRIA3GRIA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3157929-B1 PYRAZOLE COMPOUNDS AS MODULATORS OF FSHR AND USES THEREOF ARES TRADING SA (CH) 2023-12-13 EP disclosed
US-20170253605-A1 PYRAZOLE COMPOUNDS AS MODULATORS OF FSHR AND USES THEREOF TOCOPHERX, INC. (US) 2017-09-07 US disclosed
WO-2015196759-A1 PYRAZOLE COMPOUNDS AS MODULATORS OF FSHR AND USES THEREOF TOCOPHERX, INC. (US) 2015-12-30 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170253605-A1 PYRAZOLE COMPOUNDS AS MODULATORS OF FSHR AND USES THEREOF FSHR, GNRHR, LHCGR LMNA 4842/4885GRIA1 865/4885GRIA2 1313/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.