SCHEMBL17398692

SCHEMBL17398692

O=Cc1cc(C2(Cc3cccc(Cl)c3)CCCN2)cs1

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 2/20 0.38
CYP2C19 P33261 2/20 0.38
MAPT P10636 1/20 0.38
SMN1; SMN2 Q16637 2/20 0.35
CYP1A2 P05177 1/20 0.35
GAA P10253 1/20 0.35
KMT2A Q03164 3/20 0.33
DAO P14920 3/20 0.33
MEN1 O00255 2/20 0.33
ALDH1A1 P00352 1/20 0.33
HTT P42858 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
SSTR1 P30872 1/20 0.32
SSTR4 P31391 1/20 0.32
PARP1 P09874 1/20 0.32
HTR2C P28335 1/20 0.32
HTR2B P41595 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17398643 0.77 SLC6A4 (0.34) CYP2C9CYP2C19MAPTCYP1A2GAA
SCHEMBL23956497 0.77 SLC6A4 (0.34) CYP2C9CYP2C19MAPTCYP1A2GAA
SCHEMBL17428968 0.70 SLC6A4 (0.40) CYP1A2ALDH1A1
SCHEMBL29991727 0.68 PNMT (0.41) CYP2C9CYP2C19MAPTSMN1; SMN2KMT2A
SCHEMBL17398331 0.68 PNMT (0.41) CYP2C9CYP2C19MAPTSMN1; SMN2KMT2A
SCHEMBL17398398 0.68 SLC6A4 (0.35) SMN1; SMN2CYP1A2KMT2AMEN1ALDH1A1
SCHEMBL17398407 0.66 SLC6A3 (0.34) ALDH1A1
SCHEMBL17398272 0.66 SLC6A3 (0.34) ALDH1A1
SCHEMBL17398269 0.66 SLC6A3 (0.34) ALDH1A1
SCHEMBL1815990 0.65 SLC6A2 (0.46) CYP2C9CYP2C19MAPTSSTR1SSTR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3164130-A1 HETEROARYL COMPOUNDS USEFUL AS INHIBITORS OF SUMO ACTIVATING ENZYME Millennium Pharmaceuticals, Inc. (US) 2017-05-10 EP disclosed
WO-2016004136-A1 HETEROARYL COMPOUNDS USEFUL AS INHIBITORS OF SUMO ACTIVATING ENZYME DUFFEY MATTHEW O (US) 2016-01-07 WO disclosed