SCHEMBL1740260

SCHEMBL1740260

O=C(O)c1ccc(N2CCN(Cc3cnc4c(c3)NC(=O)C3CCCCN43)CC2)cc1.O=C1Nc2cc(CO)cnc2N2CCCC[C@@H]12

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 14/20 0.46
KDM4E B2RXH2 1/20 0.44
MEN1 O00255 1/20 0.44
ALDH1A1 P00352 1/20 0.44
MAPT P10636 1/20 0.44
HPGD P15428 1/20 0.44
ALOX15 P16050 1/20 0.44
KMT2A Q03164 1/20 0.44
HSD17B10 Q99714 1/20 0.44
HTR2A P28223 1/20 0.38
HTR2C P28335 1/20 0.38
HTR2B P41595 1/20 0.38
NTRK1 P04629 1/20 0.37
CRBN Q96SW2 1/20 0.36
IKZF3 Q9UKT9 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL707519 0.97 PARP1 (0.49) PARP1KDM4EMEN1ALDH1A1MAPT
SCHEMBL713960 0.97 PARP1 (0.49) PARP1KDM4EMEN1ALDH1A1MAPT
SCHEMBL709006 0.94 ALOX15 (0.50) PARP1KDM4EMEN1ALDH1A1MAPT
SCHEMBL709498 0.94 ALOX15 (0.50) PARP1KDM4EMEN1ALDH1A1MAPT
SCHEMBL1740264 0.90 PARP1 (0.45) PARP1KDM4EMEN1ALDH1A1MAPT
SCHEMBL1741938 0.87 PARP1 (0.55) PARP1KDM4EMEN1ALDH1A1MAPT
SCHEMBL707047 0.87 PARP1 (0.57) PARP1KDM4EMEN1ALDH1A1MAPT
SCHEMBL708072 0.87 ALOX15 (0.49) PARP1KDM4EMEN1ALDH1A1MAPT
SCHEMBL708071 0.87 ALOX15 (0.49) PARP1KDM4EMEN1ALDH1A1MAPT
SCHEMBL708333 0.87 PARP1 (0.48) PARP1KDM4EMEN1ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2389379-A1 Poly (ADP-Ribose) Polymerase (PARP) Inhibitors Takeda Pharmaceutical Company Limited (JP) 2011-11-30 EP disclosed