SCHEMBL17413271

SCHEMBL17413271

Cc1c(-c2cccc(Cl)c2)nc2ccccc2c1C(=O)N1CCCCCC1

nearest known ligand 0.74

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.52
KDM4E B2RXH2 2/20 0.52
TSHR P16473 1/20 0.51
PDE10A Q9Y233 1/20 0.51
DHODH Q02127 3/20 0.51
TRPV4 Q9HBA0 1/20 0.49
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
TP53 P04637 1/20 0.48
THRB P10828 1/20 0.48
NPC1 O15118 1/20 0.48
RAB9A P51151 1/20 0.48
LMNA P02545 1/20 0.48
HTT P42858 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14478824 0.88 PDE10A (0.66) TSHRPDE10ADHODHMEN1KMT2A
SCHEMBL2373562 0.83 PDE10A (0.74) MAPTKDM4ETSHRPDE10ADHODH
SCHEMBL2373101 0.79 MAPT (0.69) MAPTKDM4ETSHRPDE10ADHODH
SCHEMBL4505560 0.75 NPC1 (0.51) MAPTKDM4EMEN1KMT2ATP53
SCHEMBL4514198 0.75 NPC1 (0.51) MAPTKDM4EMEN1KMT2ATP53
SCHEMBL3322283 0.74 FABP4 (0.69) KDM4ETP53
SCHEMBL28874732 0.73 NPC1 (0.55) MAPTKDM4EMEN1KMT2ATP53
SCHEMBL4502808 0.73 NPC1 (0.50) MAPTKDM4EMEN1KMT2ATP53
SCHEMBL29387699 0.73 MAPT (0.61) MAPTKDM4ETSHRPDE10ADHODH
SCHEMBL28027244 0.72 PTGS1 (0.54) MAPTKDM4ETSHRPDE10ADHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016004035-A1 2-ARYL-4-QUINOLINECARBOXAMIDE DERIVATIVES FOR TREATING THYROID DISEASES ICAHN SCHOOL OF MEDICINE AT MOUNT SINAI (US) 2016-01-07 WO disclosed