SCHEMBL17416630

SCHEMBL17416630

COc1cc(C(=O)N(NC(C)(C)C)C(=O)c2cccc(OC(C)=O)c2C)cc(OC)c1C

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 1/20 0.46
ACHE P22303 1/20 0.37
TSHR P16473 1/20 0.37
TOP1 P11387 2/20 0.36
PKM P14618 2/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
KCNK3 O14649 1/20 0.36
KCNK9 Q9NPC2 1/20 0.36
LPAR1 Q92633 1/20 0.36
MAPK1 P28482 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7067587 0.84 ABCB1 (0.64) ABCB1NPC1RAB9AKCNK3KCNK9
SCHEMBL17416606 0.80 ABCB1 (0.56) ABCB1NPC1RAB9AKCNK3KCNK9
SCHEMBL9104050 0.80 ABCB1 (0.48) ABCB1ACHESMN1; SMN2
SCHEMBL17416628 0.80 ABCB1 (0.61) ABCB1
SCHEMBL5064249 0.80 ABCB1 (0.73) ABCB1
SCHEMBL17416624 0.76 ABCB1 (0.53) ABCB1NPC1RAB9AKCNK3KCNK9
SCHEMBL9099071 0.76 ABCB1 (0.53) ABCB1NPC1RAB9AKCNK3KCNK9
SCHEMBL9102505 0.75 ABCB1 (0.41) ABCB1TSHRNPC1RAB9ASMN1; SMN2
SCHEMBL17416625 0.75 ABCB1 (0.52) ABCB1NPC1RAB9AKCNK3KCNK9
SCHEMBL9099193 0.75 ABCB1 (0.49) ABCB1KCNK3KCNK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2460786-B1 Bioavailable diacylhydrazine ligands for modulating the expression of exogenous genes via an ecdysone receptor complex INTREXON CORP (US) 2016-01-13 EP disclosed