SCHEMBL17423643

SCHEMBL17423643

c1ccc(N2CCCNCCNCCCNCC2)cc1

nearest known ligand 0.77

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 3/20 0.77
ADRB1 P08588 3/20 0.77
HTR3E A5X5Y0 2/20 0.77
HTR3B O95264 2/20 0.77
HTR3D Q70Z44 2/20 0.77
HTR3C Q8WXA8 2/20 0.77
SIGMAR1 Q99720 2/20 0.77
CHRNB2 P17787 4/20 0.60
CHRNA4 P43681 4/20 0.60
HTR1A P08908 2/20 0.56
HTR7 P34969 2/20 0.56
LTA4H P09960 1/20 0.56
USP2 O75604 4/20 0.56
CYP2D6 P10635 3/20 0.56
ALDH1A1 P00352 3/20 0.56
TSHR P16473 2/20 0.56
CYP3A4 P08684 2/20 0.56
CYP2C19 P33261 1/20 0.56
HTR6 P50406 3/20 0.53
HSD17B10 Q99714 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3066756 0.96 ADRB1 (0.83) HTR3AADRB1HTR3EHTR3BHTR3D
SCHEMBL17431930 0.92 HTR3A (0.77) HTR3AADRB1HTR3EHTR3BHTR3D
Phenylpiperazine SCHEMBL27450129 0.90 ADRB1 (0.95) HTR3AADRB1HTR3EHTR3BHTR3D
SCHEMBL7934360 0.90 ADRB1 (0.95) HTR3AADRB1HTR3EHTR3BHTR3D
SCHEMBL17423645 0.90 ADRB1 (0.95) HTR3AADRB1HTR3EHTR3BHTR3D
Phenylpiperazine SCHEMBL3559958 0.88 ADRB1 (0.83) HTR3AADRB1HTR3EHTR3BHTR3D
Phenylpiperazine SCHEMBL29135595 0.88 ADRB1 (1.00) HTR3AADRB1HTR3EHTR3BHTR3D
Phenylpiperazine SCHEMBL24889 0.88 ADRB1 (1.00) HTR3AADRB1HTR3EHTR3BHTR3D
Phenylpiperazine SCHEMBL55125 0.88 ADRB1 (1.00) HTR3AADRB1HTR3EHTR3BHTR3D
Phenylpiperazine SCHEMBL27858598 0.88 ADRB1 (1.00) HTR3AADRB1HTR3EHTR3BHTR3D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016005892-A1 PROCESS FOR THE PREPARATION OF SUBSTITUTED POLYAZAMACROCYCLES ENI S.P.A. (IT) 2016-01-14 WO disclosed
WO-2016005892-A1 PROCESS FOR THE PREPARATION OF SUBSTITUTED POLYAZAMACROCYCLES ENI S.P.A. (IT) 2016-01-14 WO disclosed