SCHEMBL1742387

SCHEMBL1742387

NS(=O)(=O)c1cccnc1Cl

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 6/20 0.56
CA2 P00918 6/20 0.56
CA9 Q16790 2/20 0.56
MAPK1 P28482 1/20 0.56
LMNA P02545 4/20 0.54
NPSR1 Q6W5P4 1/20 0.50
NPC1 O15118 1/20 0.50
HPGD P15428 1/20 0.50
HTT P42858 1/20 0.50
KDM4E B2RXH2 1/20 0.50
MEN1 O00255 1/20 0.50
ALDH1A1 P00352 1/20 0.50
KMT2A Q03164 1/20 0.50
FTO Q9C0B1 1/20 0.47
NFE2L2 Q16236 7/20 0.46
CA4 P22748 2/20 0.43
CA6 P23280 2/20 0.43
CA12 O43570 1/20 0.43
CYP2C9 P11712 1/20 0.43
CA5A P35218 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29435677 0.81 TRPV4 (0.51) CA1CA2CA9MAPK1LMNA
SCHEMBL349118 0.81 TRPV4 (0.51) CA1CA2CA9MAPK1LMNA
SCHEMBL31634218 0.79 NFE2L2 (0.46) CA1CA2CA9MAPK1LMNA
SCHEMBL3704196 0.79 COMT (0.47) LMNANPC1HPGDHTTMEN1
SCHEMBL925929 0.79 NFE2L2 (0.46) CA1CA2CA9MAPK1LMNA
SCHEMBL3698654 0.78 COMT (0.46) LMNANPC1HPGDHTTMEN1
SCHEMBL3698653 0.78 NFE2L2 (0.45) CA1CA2CA9MAPK1LMNA
Lithium Ion SCHEMBL3698633 0.78 NFE2L2 (0.45) CA1CA2CA9MAPK1LMNA
SCHEMBL3698635 0.78 COMT (0.46) LMNANPC1HPGDHTTMEN1
SCHEMBL3713453 0.78 COMT (0.46) LMNANPC1HPGDHTTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 82 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024115549-A1 ARYL- AND HETEROARYL-SULFONAMIDE DERIVATIVES AS CCR8 MODULATORS IDORSIA PHARMACEUTICALS LTD (CH) 2024-06-06 WO claimed
EP-0131861-A2 2-Substituted-3-sulfonamidepyridine compounds, process for preparing and pharmaceutical compositions comprising the same FABRICA DE PRODUCTOS QUIMICOS Y FARMACEUTICOS ABELLO, S.A. (ES) 1985-01-23 EP claimed
WO-2024115549-A1 ARYL- AND HETEROARYL-SULFONAMIDE DERIVATIVES AS CCR8 MODULATORS IDORSIA PHARMACEUTICALS LTD (CH) 2024-06-06 WO disclosed
US-20210380548-A1 Fused [1,2,4]Thiadiazine Derivatives Which Act as KAT Inhibitors of the MYST Family CTXT PTY LIMITED (AU) 2021-12-09 US disclosed
US-20210380548-A1 Fused [1,2,4]Thiadiazine Derivatives Which Act as KAT Inhibitors of the MYST Family CTXT PTY LIMITED (AU) 2021-12-09 US disclosed
US-10844013-B2 Phenyl amino piperidine mTORC inhibitors and uses thereof NAVITOR PHARMACEUTICALS, INC. (US) 2020-11-24 US disclosed
US-10844013-B2 Phenyl amino piperidine mTORC inhibitors and uses thereof NAVITOR PHARMACEUTICALS, INC. (US) 2020-11-24 US disclosed
EP-3676266-A1 FUSED [1,2,4]THIADIAZINE DERIVATIVES WHICH ACT AS KAT INHIBITORS OF THE MYST FAMILY Ctxt Pty Ltd (AU) 2020-07-08 EP disclosed
US-20200207716-A1 PHENYL AMINO PIPERIDINE mTORC INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. 2020-07-02 US disclosed
US-20200207716-A1 PHENYL AMINO PIPERIDINE mTORC INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. 2020-07-02 US disclosed
EP-3538091-A1 PHENYL AMINO PIPERIDINE mTORC INHIBITORS AND USES THEREOF Navitor Pharmaceuticals, Inc. (US) 2019-09-18 EP disclosed
US-4690707-A PRE- AND POSTEMERGENCE HERBICIDES; PLANT GROWTH REGULATORS; PREFERENTIAL CIBA-GEIGY CORPORATION (US) 1987-09-01 US disclosed
US-4657578-A Herbicidal ortho-heterocyclic sulfonamides E. I. DU PONT DE NEMOURS AND COMPANY (US) 1987-04-14 US disclosed
US-4643760-A Herbicidal sulfonylureas CIBA-GEIGY CORPORATION (US) 1987-02-17 US disclosed
EP-0178101-A1 Herbicidal ortho-heterocyclic sulfonamides E.I. DU PONT DE NEMOURS AND COMPANY (US) 1986-04-16 EP disclosed
US-4579583-A HERBICIDES, GROWTH REGULATORS CIBA-GEIGY CORPORATION (US) 1986-04-01 US disclosed
US-4549898-A PREEMERGENT AND POSTEMERGENT HERBICIDES CIBA-GEIGY CORPORATION (US) 1985-10-29 US disclosed
EP-0145664-A2 Herbicidal sulfonyl ureas CIBA-GEIGY AG (CH) 1985-06-19 EP disclosed
EP-0103543-A2 Sulfonyl ureas CIBA-GEIGY AG (CH) 1984-03-21 EP disclosed
EP-0097122-A2 N-heterocyclosulfonyl-N'-pyrimidinyl and triazinyl ureas CIBA-GEIGY AG (CH) 1983-12-28 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210380548-A1 Fused [1,2,4]Thiadiazine Derivatives Which Act as KAT Inhibitors of the MYST Family KAT5, KAT6A, KAT2A CA1 3478/4885CA2 4004/4885CA9 4651/4885
US-10844013-B2 Phenyl amino piperidine mTORC inhibitors and uses thereof MTOR, RICTOR, RPTOR CA1 4540/4885CA2 3770/4885CA9 4552/4885
US-20200207716-A1 PHENYL AMINO PIPERIDINE mTORC INHIBITORS AND USES THEREOF MTOR, RICTOR, RPTOR CA1 4540/4885CA2 3770/4885CA9 4552/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.