SCHEMBL174328

SCHEMBL174328

CC(C)(C)c1ccc(Nc2ccc(-c3noc(C4CCC(C(=O)O)CC4)n3)cc2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR4 O95977 2/20 0.49
S1PR1 P21453 2/20 0.49
S1PR5 Q9H228 2/20 0.49
S1PR3 Q99500 1/20 0.49
GAA P10253 2/20 0.46
KDM4E B2RXH2 2/20 0.46
CA12 O43570 1/20 0.45
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45
CA9 Q16790 1/20 0.45
SMN1; SMN2 Q16637 8/20 0.44
LMNA P02545 4/20 0.44
HTT P42858 3/20 0.44
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
TP53 P04637 4/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
MAPT P10636 5/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL174317 1.00 S1PR4 (0.49) S1PR4S1PR1S1PR5S1PR3GAA
SCHEMBL162177 0.91 S1PR4 (0.49) S1PR4S1PR1S1PR5S1PR3GAA
SCHEMBL174329 0.91 S1PR4 (0.49) S1PR4S1PR1S1PR5S1PR3GAA
SCHEMBL6370573 0.82 RAB9A (0.60) GAAKDM4ECA12CA1CA2
SCHEMBL161998 0.80 NPC1 (0.56) GAAKDM4ECA12CA1CA2
SCHEMBL162121 0.80 NPC1 (0.56) GAAKDM4ECA12CA1CA2
SCHEMBL15021866 0.79 HDAC4 (0.51) S1PR4S1PR1S1PR5GAAKDM4E
SCHEMBL174631 0.79 KMT2A (0.50) CA12CA1CA2CA9LMNA
SCHEMBL163930 0.79 HDAC4 (0.51) S1PR4S1PR1S1PR5GAAKDM4E
SCHEMBL171022 0.78 CA12 (0.56) S1PR1S1PR5CA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2611783-A2 HETEROCYCLIC COMPOUNDS AS DGAT1 INHIBITORS Piramal Enterprises Limited (IN) 2013-07-10 EP disclosed
WO-2012029032-A2 HETEROCYCLIC COMPOUNDS AS DGAT1 INHIBITORS PIRAMAL LIFE SCIENCES LIMITED (IN) 2012-03-08 WO disclosed