SCHEMBL17445832

SCHEMBL17445832

COC(=O)/C=C/CNC(=O)c1cc(C)n(Cc2ccco2)c1C

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 14/20 0.55
POLB P06746 9/20 0.55
HTT P42858 2/20 0.55
GAA P10253 2/20 0.55
MAPT P10636 2/20 0.55
KLKB1 P03952 1/20 0.55
MEN1 O00255 4/20 0.53
KMT2A Q03164 4/20 0.53
RECQL P46063 2/20 0.53
RAB9A P51151 11/20 0.52
NPC1 O15118 9/20 0.52
TDP1 Q9NUW8 3/20 0.51
SMN1; SMN2 Q16637 6/20 0.49
KDM4E B2RXH2 3/20 0.49
PKM P14618 1/20 0.48
TSHR P16473 3/20 0.48
L3MBTL1 Q9Y468 2/20 0.46
HPGD P15428 1/20 0.46
ALOX15 P16050 1/20 0.46
HSD17B10 Q99714 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30475627 0.75 ALDH1A1 (0.74) ALDH1A1POLBHTTGAAMAPT
SCHEMBL25062631 0.73 ALDH1A1 (0.63) ALDH1A1POLBHTTGAAMAPT
SCHEMBL554044 0.71 KLKB1 (1.00) ALDH1A1POLBHTTGAAMAPT
SCHEMBL25062623 0.70 ALDH1A1 (0.62) ALDH1A1POLBHTTGAAMAPT
SCHEMBL24554002 0.66 ALDH1A1 (0.56) ALDH1A1POLBHTTGAAMAPT
SCHEMBL17445810 0.66 KMT2A (0.41) ALDH1A1POLBGAAMAPTMEN1
SCHEMBL17445842 0.66 ALDH1A1 (0.50) ALDH1A1POLBGAAMAPTMEN1
SCHEMBL17445835 0.65 KDM4E (0.53) ALDH1A1MAPTMEN1KMT2ARECQL
SCHEMBL17445800 0.65 HPGD (0.49) ALDH1A1POLBHTTGAAMAPT
SCHEMBL17447416 0.63 ALDH1A1 (0.47) ALDH1A1GAAMEN1KMT2ARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10273208-B2 Screening methods for the binding affinity of chemical entities to biological molecules and NEDD4-1 inhibitors identified by the screening methods NORTHWESTERN UNIVERSITY (US) 2019-04-30 US disclosed
US-20170152228-A1 SCREENING METHODS FOR THE BINDING AFFINITY OF CHEMICAL ENTITIES TO BIOLOGICAL MOLECULES AND NEDD4-1 INHIBITORS IDENTIFIED BY THE SCREENING METHODS NORTHWESTERN UNIVERSITY (US) 2017-06-01 US disclosed
US-20170152228-A1 SCREENING METHODS FOR THE BINDING AFFINITY OF CHEMICAL ENTITIES TO BIOLOGICAL MOLECULES AND NEDD4-1 INHIBITORS IDENTIFIED BY THE SCREENING METHODS NORTHWESTERN UNIVERSITY (US) 2017-06-01 US disclosed
US-9586890-B2 Screening methods for the binding affinity of chemical entities to biological molecules and NEDD4-1 inhibitors identified by the screening methods NORTHWESTERN UNIVERSITY (US) 2017-03-07 US disclosed
US-9586890-B2 Screening methods for the binding affinity of chemical entities to biological molecules and NEDD4-1 inhibitors identified by the screening methods NORTHWESTERN UNIVERSITY (US) 2017-03-07 US disclosed
US-20160016893-A1 SCREENING METHODS FOR THE BINDING AFFINITY OF CHEMICAL ENTITIES TO BIOLOGICAL MOLECULES AND NEDD4-1 INHIBITORS IDENTIFIED BY THE SCREENING METHODS NORTHWESTERN UNIVERSITY (US) 2016-01-21 US disclosed
US-20160016893-A1 SCREENING METHODS FOR THE BINDING AFFINITY OF CHEMICAL ENTITIES TO BIOLOGICAL MOLECULES AND NEDD4-1 INHIBITORS IDENTIFIED BY THE SCREENING METHODS NORTHWESTERN UNIVERSITY (US) 2016-01-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170152228-A1 SCREENING METHODS FOR THE BINDING AFFINITY OF CHEMICAL ENTITIES TO BIOLOGICAL MOLECULES AND NEDD4-1 INHIBITORS IDENTIFIED BY THE SCREENING METHODS NEDD4, STUB1, CUL1 ALDH1A1 1314/4885POLB 3357/4885HTT 3191/4885
US-20160016893-A1 SCREENING METHODS FOR THE BINDING AFFINITY OF CHEMICAL ENTITIES TO BIOLOGICAL MOLECULES AND NEDD4-1 INHIBITORS IDENTIFIED BY THE SCREENING METHODS NEDD4, STUB1, UBQLN1 ALDH1A1 2967/4885POLB 3390/4885HTT 1034/4885
US-10273208-B2 Screening methods for the binding affinity of chemical entities to biological molecules and NEDD4-1 inhibitors identified by the screening methods NEDD4, STUB1, CUL1 ALDH1A1 1314/4885POLB 3357/4885HTT 3191/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.