SCHEMBL1744814

SCHEMBL1744814

O=C1CCc2cc(CBr)[c]cc2N1

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.40
MAPK13 O15264 1/20 0.40
MAPK12 P53778 1/20 0.40
MAPK11 Q15759 1/20 0.40
MAPK14 Q16539 1/20 0.40
CA9 Q16790 1/20 0.39
KIF11 P52732 3/20 0.37
MAOA P21397 10/20 0.37
MAOB P27338 10/20 0.37
CYP11B1 P15538 3/20 0.36
CYP11B2 P19099 3/20 0.36
CYP19A1 P11511 2/20 0.36
PDE3B Q13370 3/20 0.35
PDE3A Q14432 3/20 0.35
TBXAS1 P24557 2/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2C9 P11712 1/20 0.35
CRBN Q96SW2 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1744197 0.78 NPC1 (0.43) NPC1MAPK13MAPK12MAPK11MAPK14
SCHEMBL9435206 0.71 CA9 (0.42) NPC1MAPK13MAPK12MAPK11MAPK14
SCHEMBL14796816 0.70 MAOA (0.51) NPC1MAPK13MAPK12MAPK11MAPK14
SCHEMBL14843503 0.67 CA9 (0.57) NPC1MAPK13MAPK12MAPK11MAPK14
SCHEMBL29754233 0.67 CA9 (0.57) NPC1MAPK13MAPK12MAPK11MAPK14
SCHEMBL6217777 0.65 MAOA (0.50) NPC1MAPK13MAPK12MAPK11MAPK14
SCHEMBL910409 0.63 NPC1 (0.55) NPC1MAPK13MAPK12MAPK11MAPK14
SCHEMBL99208 0.63 MAOA (0.56) NPC1MAPK13MAPK12MAPK11MAPK14
SCHEMBL12682656 0.62 CYP11B1 (0.56) NPC1MAPK13MAPK12MAPK11MAPK14
SCHEMBL19278654 0.62 CA9 (0.52) NPC1MAPK13MAPK12MAPK11MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2385939-A1 DIHYDROPYRIDONE AMIDES AS P2X7 MODULATORS F. Hoffmann-La Roche AG (CH) 2011-11-16 EP disclosed
US-8041551-B1 Algorithm and architecture for multi-argument associative operations that minimizes the number of components using a latency of the components THE MATHWORKS, INC. (US) 2011-10-18 US disclosed
WO-2010072597-A1 DIHYDROPYRIDONE AMIDES AS P2X7 MODULATORS F. HOFFMANN-LA ROCHE AG (CH) 2010-07-01 WO disclosed