SCHEMBL17450128

SCHEMBL17450128

CCn1cnc2c(NCc3ccccc3)nc(F)nc21

nearest known ligand 0.60

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 6/20 0.60
CTSL P07711 5/20 0.55
TMIGD3 P0DMS9 2/20 0.55
ADORA2A P29274 2/20 0.55
ADORA1 P30542 2/20 0.55
CDK5 Q00535 1/20 0.54
KDM4E B2RXH2 1/20 0.52
NPC1 O15118 1/20 0.52
MAPT P10636 1/20 0.52
TDP1 Q9NUW8 1/20 0.52
ADORA2B P29275 1/20 0.52
CDK2 P24941 2/20 0.52
CCNA2 P20248 1/20 0.52
CCNA1 P78396 1/20 0.52
CACNA1B Q00975 1/20 0.52
YTHDC1 Q96MU7 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17450223 0.88 CDK1 (0.60) CDK1CTSLTMIGD3ADORA2AADORA1
SCHEMBL17450142 0.87 CTSL (0.67) CDK1CTSLTMIGD3ADORA2AADORA1
SCHEMBL17450224 0.87 CDK1 (0.57) CDK1CTSLTMIGD3ADORA2AADORA1
SCHEMBL17450179 0.86 CDK1 (0.56) CDK1CTSLTMIGD3ADORA2AADORA1
SCHEMBL17450124 0.85 CDK1 (0.72) CDK1CTSLTMIGD3ADORA2AADORA1
SCHEMBL20350685 0.85 CDK1 (0.73) CDK1CTSLTMIGD3ADORA2AADORA1
SCHEMBL17442999 0.85 CDK1 (0.73) CDK1CDK5KDM4ENPC1MAPT
SCHEMBL17450131 0.82 CTSL (0.72) CDK1CTSLCDK2YTHDC1
SCHEMBL21609988 0.81 CDK1 (0.53) CDK1CTSLTMIGD3ADORA2AADORA1
SCHEMBL3851604 0.81 TDP1 (0.78) CDK1CDK5KDM4ENPC1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016011394-A1 IMAGING AGENTS FOR NEURAL FLUX THE GENERAL HOSPITAL CORPORATION (US) 2016-01-21 WO disclosed