Alpha-Ketoglutaric Acid

Alpha-Ketoglutaric Acid

SCHEMBL174620

ClCc1ccc2c(c1)CCNCC2.O=C(O)CCC(=O)C(=O)O

nearest known ligand 0.43

Full drug profile on Sugi Atlas →

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MLNR O43193 8/20 0.43
CYP2D6 P10635 2/20 0.40
HTR2C P28335 3/20 0.40
HTR2B P41595 2/20 0.40
HTR2A P28223 1/20 0.40
ACHE P22303 1/20 0.39
ALDH1A1 P00352 1/20 0.38
DRD2 P14416 1/20 0.38
DRD1 P21728 1/20 0.38
ITGB3 P05106 1/20 0.37
ITGA2B P08514 1/20 0.37
MAPK1 P28482 1/20 0.37
SLC13A3 Q8WWT9 1/20 0.37
EGLN1 Q9GZT9 1/20 0.37
OR51E2 Q9H255 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Succinic Acid SCHEMBL174914 0.93 HTR2C (0.45) MLNRCYP2D6HTR2CHTR2BHTR2A
Adipic Acid SCHEMBL173690 0.88 HTR2C (0.42) MLNRCYP2D6HTR2CHTR2BHTR2A
Malonic Acid SCHEMBL173339 0.85 HTR2C (0.45) MLNRCYP2D6HTR2CHTR2BHTR2A
Glycolic Acid SCHEMBL174349 0.85 HTR2C (0.45) MLNRCYP2D6HTR2CHTR2BHTR2A
SCHEMBL162032 0.81 HTR2C (0.57) MLNRCYP2D6HTR2CHTR2BHTR2A
Glutamic Acid SCHEMBL175044 0.80 GRIK1 (0.43) MLNRCYP2D6HTR2CHTR2BHTR2A
Alpha-Ketoglutaric Acid SCHEMBL16464850 0.80 HTR2C (0.53) HTR2CHTR2BALDH1A1DRD2DRD1
Bromide SCHEMBL174563 0.80 HTR2C (0.55) MLNRCYP2D6HTR2CHTR2BHTR2A
Nitric Acid SCHEMBL174071 0.79 MLNR (0.47) MLNRCYP2D6HTR2CHTR2BHTR2A
Phosphoric Acid SCHEMBL174207 0.79 HTR2C (0.47) MLNRCYP2D6HTR2CHTR2BHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2611449-A1 ADMINISTRATION OF LORCASERIN TO INDIVIDUALS WITH RENAL IMPAIRMENT Arena Pharmaceuticals, Inc. (US) 2013-07-10 EP disclosed
WO-2012030939-A1 ADMINISTRATION OF LORCASERIN TO INDIVIDUALS WITH RENAL IMPAIRMENT ARENA PHARMACEUTICALS, INC. (US) 2012-03-08 WO disclosed