SCHEMBL1746476

SCHEMBL1746476

CSc1cc(-c2ccncc2)nc2c1C(=O)N(C(=O)O)CC2

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 1/20 0.37
GSK3B P49841 6/20 0.35
HTR2A P28223 1/20 0.35
HTR2C P28335 1/20 0.35
HTR2B P41595 1/20 0.35
CYP2C9 P11712 1/20 0.34
PDE4B Q07343 5/20 0.34
BUB1 O43683 1/20 0.33
LMNA P02545 1/20 0.33
MAPK1 P28482 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2D6 P10635 1/20 0.33
GRM5 P41594 1/20 0.32
ALDH1A1 P00352 1/20 0.32
NPC1 O15118 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1746373 0.91 PDE4B (0.39) GSK3BCYP2C9PDE4BCYP1A2ALDH1A1
SCHEMBL8443924 0.78 BUB1 (0.44) PDE4BBUB1
SCHEMBL1746587 0.72 PDE4B (0.39) CYP2C9PDE4BLMNAMAPK1CYP1A2
SCHEMBL8442662 0.72 BUB1 (0.37) CYP2C9PDE4BBUB1CYP1A2ALDH1A1
SCHEMBL8442660 0.70 USP30 (0.39) PDE4BBUB1
SCHEMBL8446562 0.70 PDE4B (0.41) PDE4BBUB1LMNAALDH1A1
SCHEMBL1746280 0.69 ADORA1 (0.38) GSK3BCYP2C9PDE4BLMNAMAPK1
SCHEMBL19664854 0.64 KMO (0.42) MAPK1ALDH1A1NPC1
SCHEMBL17847603 0.63 BUB1 (0.50) BUB1
SCHEMBL19714885 0.62 CDC7 (0.64) AKT1GSK3BMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2380890-A1 New 7,8-dihydro-1,6-naphthyridin-5(6h)-one-derivatives as PDE4 inhibitors Almirall, S.A. (ES) 2011-10-26 EP disclosed
US-20110253549-A1 WASHING APPARATUS AND METHOD OF DEODORIZING WASHING WATER KANNO MINORU 2011-10-20 US disclosed