SCHEMBL1746587

SCHEMBL1746587

CS(=O)(=O)c1cc(-c2ccccc2)nc2c1C(=O)N(C(=O)O)CC2

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 4/20 0.39
BPTF Q12830 1/20 0.36
VCP P55072 2/20 0.35
USP30 Q70CQ3 1/20 0.35
POLB P06746 2/20 0.35
HSD17B10 Q99714 2/20 0.35
LMNA P02545 2/20 0.35
HPGD P15428 2/20 0.35
HTT P42858 2/20 0.35
KMT2A Q03164 2/20 0.35
NPSR1 Q6W5P4 2/20 0.35
RAB9A P51151 2/20 0.35
MEN1 O00255 1/20 0.35
S1PR4 O95977 1/20 0.35
TP53 P04637 1/20 0.35
S1PR1 P21453 1/20 0.35
SDHB P21912 1/20 0.35
MAPK1 P28482 1/20 0.35
STAT3 P40763 1/20 0.35
STAT1 P42224 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1747649 0.90 POLB (0.39) PDE4BPOLBLMNAHTTKMT2A
SCHEMBL1746282 0.88 PDE4B (0.35) PDE4B
SCHEMBL1746227 0.88 PDE4B (0.43) PDE4BVCPHSD17B10LMNAKMT2A
SCHEMBL8446595 0.87 BUB1 (0.44) PDE4BUSP30ACACBACACA
SCHEMBL1747642 0.84 NPSR1 (0.41) PDE4BVCPHSD17B10LMNAHPGD
SCHEMBL1746373 0.81 PDE4B (0.39) PDE4BUSP30POLBHSD17B10HTT
SCHEMBL1747304 0.78 LMNA (0.35) PDE4BBPTFVCPPOLBHSD17B10
SCHEMBL8443971 0.77 USP30 (0.38) PDE4BUSP30POLBKMT2AMEN1
SCHEMBL8442707 0.77 PDE4B (0.41) PDE4BUSP30HSD17B10HPGDKMT2A
SCHEMBL8443926 0.76 GPR119 (0.37) PDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2380890-A1 New 7,8-dihydro-1,6-naphthyridin-5(6h)-one-derivatives as PDE4 inhibitors Almirall, S.A. (ES) 2011-10-26 EP disclosed
US-20110253549-A1 WASHING APPARATUS AND METHOD OF DEODORIZING WASHING WATER KANNO MINORU 2011-10-20 US disclosed