SCHEMBL1746529

SCHEMBL1746529

CSc1cc(-c2ccccc2)nc2c1C(=O)N(C(=O)O)CC2C

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 5/20 0.38
ADORA2A P29274 3/20 0.38
CYP2C9 P11712 1/20 0.36
KDM4E B2RXH2 3/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
GSK3B P49841 1/20 0.35
POLB P06746 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
PDE4B Q07343 1/20 0.35
ALDH1A1 P00352 3/20 0.33
MAPK1 P28482 1/20 0.33
ADORA3 P0DMS8 3/20 0.33
TSHR P16473 1/20 0.33
LMNA P02545 1/20 0.32
HPGD P15428 1/20 0.32
HTT P42858 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
TDP1 Q9NUW8 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1746373 0.77 PDE4B (0.39) ADORA1ADORA2ACYP2C9KDM4EMEN1
SCHEMBL1747614 0.68 POLB (0.39) ADORA1ADORA2AKDM4EMEN1KMT2A
SCHEMBL8443924 0.68 BUB1 (0.44) ADORA1ADORA2APDE4B
SCHEMBL8445470 0.67 ABCB1 (0.36) ADORA1ADORA2APDE4BALDH1A1MAPK1
SCHEMBL1746137 0.60 TSHR (0.48) CYP2C9MEN1KMT2APOLBPDE4B
SCHEMBL28020209 0.56 TSHR (0.43) ADORA1ADORA2AKDM4EMEN1KMT2A
SCHEMBL1735055 0.56 MCL1 (0.50) ADORA1KDM4EMEN1KMT2ASMN1; SMN2
SCHEMBL13133556 0.56 MAPT (0.58) ADORA1ADORA2AKDM4EMEN1KMT2A
SCHEMBL9619520 0.56 MEN1 (0.50) ADORA1ADORA2AKDM4EMEN1KMT2A
SCHEMBL1733453 0.55 KDM4E (0.57) CYP2C9KDM4EMEN1KMT2APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2380890-A1 New 7,8-dihydro-1,6-naphthyridin-5(6h)-one-derivatives as PDE4 inhibitors Almirall, S.A. (ES) 2011-10-26 EP disclosed
US-20110253549-A1 WASHING APPARATUS AND METHOD OF DEODORIZING WASHING WATER KANNO MINORU 2011-10-20 US disclosed