SCHEMBL1746545

SCHEMBL1746545

Cc1ccc(C(=O)NC2CC2)cc1-c1cccc(-c2cc(N)c3c(n2)CCNC3=O)c1

nearest known ligand 0.56

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 8/20 0.56
MAPK14 Q16539 12/20 0.51
LCK P06239 2/20 0.49
KDR P35968 2/20 0.49
CSF1R P07333 1/20 0.49
KIT P10721 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1747651 0.89 PDE4B (0.65) PDE4BMAPK14
SCHEMBL1746553 0.88 PDE4B (0.52) PDE4BMAPK14
SCHEMBL1746258 0.82 PDE4B (0.84) PDE4BMAPK14
SCHEMBL1747376 0.73 PDE4B (0.73) PDE4B
SCHEMBL1746589 0.72 PDE4B (1.00) PDE4B
SCHEMBL1746610 0.71 PDE4B (0.78) PDE4B
SCHEMBL1746288 0.70 PDE4B (1.00) PDE4B
SCHEMBL1747621 0.70 PDE4B (1.00) PDE4B
SCHEMBL31367847 0.70 MAPK14 (0.74) MAPK14LCKKDRCSF1RKIT
SCHEMBL1746325 0.68 PDE4B (0.73) PDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2380890-A1 New 7,8-dihydro-1,6-naphthyridin-5(6h)-one-derivatives as PDE4 inhibitors Almirall, S.A. (ES) 2011-10-26 EP disclosed
EP-2380890-A1 New 7,8-dihydro-1,6-naphthyridin-5(6h)-one-derivatives as PDE4 inhibitors Almirall, S.A. (ES) 2011-10-26 EP disclosed
US-20110253549-A1 WASHING APPARATUS AND METHOD OF DEODORIZING WASHING WATER KANNO MINORU 2011-10-20 US disclosed