SCHEMBL17469676

SCHEMBL17469676

CCCCOc1cc(OC)cc2c1C(=O)c1c(O)ccc(OC)c1C2

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.40
CNR2 P34972 1/20 0.39
ELANE P08246 1/20 0.39
CYSLTR2 Q9NS75 1/20 0.39
CYSLTR1 Q9Y271 1/20 0.39
THRA P10827 2/20 0.38
THRB P10828 2/20 0.38
LMNA P02545 1/20 0.38
TSHR P16473 1/20 0.38
HTT P42858 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA4 P22748 1/20 0.37
CA6 P23280 1/20 0.37
PDE4A P27815 1/20 0.36
PDE4B Q07343 1/20 0.36
PDE4C Q08493 1/20 0.36
PDE4D Q08499 1/20 0.36
AHR P35869 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19476034 0.89 CES2 (0.38) CES2CNR2ELANECYSLTR2CYSLTR1
SCHEMBL19476243 0.86 CYSLTR2 (0.37) CES2CNR2ELANECYSLTR2CYSLTR1
SCHEMBL19476244 0.84 PSEN1 (0.46)
SCHEMBL19476058 0.83 KDM4E (0.40) CES2CA1CA2CA4CA6
SCHEMBL19175928 0.83 CA1 (0.45) SMN1; SMN2CA1CA2CA4CA6
SCHEMBL19476170 0.82 KDM4E (0.47) CES2ELANETHRBTSHRSMN1; SMN2
SCHEMBL19476060 0.79 MAOB (0.39)
SCHEMBL19476171 0.78 PARP15 (0.46) LMNAHTTCA1CA2CA4
SCHEMBL19168589 0.73 NPC1 (0.40) SMN1; SMN2PDE4APDE4BPDE4CPDE4D
SCHEMBL19476241 0.73 CA1 (0.39) SMN1; SMN2CA1CA2ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017180248-A1 ENANTIOENRICHED VIRIDICATUMTOXIN B ANALOGS WILLIAM MARSH RICE UNIVERSITY (US) 2017-10-19 WO disclosed
US-20170210699-A1 PREPARATION AND BIOLOGICAL EVALUATION OF VIRIDICATUMTOXIN ANALOGS WILLIAM MARSH RICE UNIVERSITY (US) 2017-07-27 US disclosed
WO-2016014643-A1 PREPARATION AND BIOLOGICAL EVALUATION OF VIRIDICATUMTOXIN ANALOGS WILLIAM MARSH RICE UNIVERSITY (US) 2016-01-28 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170210699-A1 PREPARATION AND BIOLOGICAL EVALUATION OF VIRIDICATUMTOXIN ANALOGS VIP, DDOST, ANTXR2 CES2 3385/4885CNR2 4401/4885ELANE 499/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.