SCHEMBL19476171

SCHEMBL19476171

COc1cc2c(c(OCc3cccc4ccccc34)c1)C(=O)c1c(O)ccc(OC)c1C2

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP15 Q460N3 1/20 0.46
PARP10 Q53GL7 1/20 0.46
CETP P11597 1/20 0.42
AKR1B1 P15121 2/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA4 P22748 1/20 0.41
CA6 P23280 1/20 0.41
KEAP1 Q14145 1/20 0.40
NFE2L2 Q16236 1/20 0.40
KDM4E B2RXH2 2/20 0.40
ALDH1A1 P00352 1/20 0.40
MEN1 O00255 4/20 0.38
KMT2A Q03164 4/20 0.38
HSP90AA1 P07900 1/20 0.37
HSP90AB1 P08238 1/20 0.37
MCL1 Q07820 1/20 0.37
P2RY12 Q9H244 1/20 0.36
FFAR1 O14842 1/20 0.36
LMNA P02545 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19175928 0.84 CA1 (0.45) CA1CA2CA4CA6ALDH1A1
SCHEMBL19476025 0.80 PARP10 (0.47) PARP15PARP10AKR1B1CA1CA2
SCHEMBL19476170 0.78 KDM4E (0.47) CA1CA2CA4CA6KDM4E
SCHEMBL17469676 0.78 CES2 (0.40) CA1CA2CA4CA6LMNA
SCHEMBL19476058 0.77 KDM4E (0.40) CA1CA2CA4CA6KDM4E
SCHEMBL19476060 0.76 MAOB (0.39) MEN1KMT2AFFAR1
SCHEMBL19168589 0.75 NPC1 (0.40) ALDH1A1MEN1KMT2AMAPT
SCHEMBL19476241 0.75 CA1 (0.39) CA1CA2
SCHEMBL19476035 0.75 CA1 (0.39) CA1CA2
SCHEMBL19476245 0.74 PSEN1 (0.42) CA1CA2KEAP1NFE2L2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017180248-A1 ENANTIOENRICHED VIRIDICATUMTOXIN B ANALOGS WILLIAM MARSH RICE UNIVERSITY (US) 2017-10-19 WO disclosed