SCHEMBL17478147

SCHEMBL17478147

CC1=C(C(=O)O)C(c2ccc(C(F)(F)F)nc2)CC(=O)N1

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 4/20 0.47
LMNA P02545 1/20 0.46
HTT P42858 1/20 0.44
ROCK1 Q13464 8/20 0.44
RPS6KA1 Q15418 7/20 0.44
RPS6KB1 P23443 6/20 0.43
ROCK2 O75116 1/20 0.43
HDAC4 P56524 1/20 0.40
TP53 P04637 3/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17484775 0.87 HTT (0.62) GPBAR1LMNAHTTROCK1RPS6KA1
SCHEMBL17478177 0.87 HTT (0.62) GPBAR1LMNAHTTROCK1RPS6KA1
SCHEMBL17478072 0.81 LMNA (0.49) GPBAR1LMNAHTTROCK1RPS6KA1
SCHEMBL3895930 0.81 GPBAR1 (0.67) GPBAR1LMNAHTTROCK1RPS6KA1
SCHEMBL3342133 0.77 LMNA (0.58) GPBAR1LMNAHTTROCK1RPS6KA1
SCHEMBL3888823 0.74 GPBAR1 (0.65) GPBAR1LMNAHTTTP53
SCHEMBL5661329 0.74 ADRA1A (0.52) GPBAR1LMNAHTTTP53
SCHEMBL7928701 0.74 ADRA1A (0.52) GPBAR1LMNAHTTTP53
SCHEMBL17478253 0.72 RPS6KB1 (0.55) GPBAR1LMNAHTTROCK1RPS6KA1
SCHEMBL4312703 0.70 RPS6KB1 (0.58) GPBAR1LMNAHTTROCK1RPS6KA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3174872-A1 2-OXO-3,4-DIHYDROPYRIDINE-5-CARBOXYLATES AND THEIR USE Université de Lille 2 Droit et Santé (FR) 2017-06-07 EP disclosed
WO-2016016238-A1 2-OXO-3,4-DIHYDROPYRIDINE-5-CARBOXYLATES AND THEIR USE UNIVERSITE DE LILLE 2 DROIT ET SANTE (FR) 2016-02-04 WO disclosed