SCHEMBL17479481

SCHEMBL17479481

CC(=O)c1ccc(OC(N)=O)cc1Cl

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.48
MEN1 O00255 1/20 0.48
ALDH1A1 P00352 2/20 0.42
MAPK1 P28482 2/20 0.42
CYP3A4 P08684 1/20 0.42
HPGD P15428 1/20 0.42
JAK2 O60674 1/20 0.41
TYK2 P29597 1/20 0.41
NR1H4 Q96RI1 2/20 0.41
MAOA P21397 3/20 0.40
MAOB P27338 3/20 0.40
KDM4E B2RXH2 2/20 0.40
MAPT P10636 4/20 0.40
RAB9A P51151 2/20 0.40
GABRA1 P14867 3/20 0.38
GABRG2 P18507 3/20 0.38
GABRB3 P28472 3/20 0.38
GABRB2 P47870 2/20 0.38
NPC1 O15118 1/20 0.38
CASP3 P42574 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17479464 0.81 KMT2A (0.50) KMT2AMEN1ALDH1A1MAPK1CYP3A4
SCHEMBL473972 0.80 ALDH1A1 (0.65) KMT2AMEN1ALDH1A1MAPK1CYP3A4
SCHEMBL23753577 0.80 MEN1 (0.57) KMT2AMEN1ALDH1A1CYP3A4KDM4E
SCHEMBL17479453 0.79 MAOB (0.54) KMT2AMEN1ALDH1A1MAPK1CYP3A4
SCHEMBL18758272 0.79 ALDH1A1 (0.44) KMT2AALDH1A1MAPK1CYP3A4HPGD
SCHEMBL7170047 0.79 MEN1 (0.52) KMT2AMEN1ALDH1A1MAPK1CYP3A4
SCHEMBL31266502 0.79 MEN1 (0.52) KMT2AMEN1ALDH1A1MAPK1CYP3A4
SCHEMBL29042305 0.78 KMT2A (0.43) KMT2AMEN1ALDH1A1MAPK1HPGD
SCHEMBL22406996 0.77 HSP90AA1 (0.53) KMT2AMEN1ALDH1A1MAPK1CYP3A4
SCHEMBL17242255 0.77 MEN1 (0.53) KMT2AMEN1ALDH1A1NR1H4MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3180317-A1 FACTOR XIa INHIBITORS Merck Sharp & Dohme Corp. (US) 2017-06-21 EP disclosed
WO-2016015593-A1 FACTOR XIa INHIBITORS MERCK SHARP & DOHME CORP. (US) 2016-02-04 WO disclosed