SCHEMBL17479554

SCHEMBL17479554

[2H]C([2H])([2H])NC(=O)Oc1ccc(C(C)=O)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.52
RAB9A P51151 2/20 0.52
HPGD P15428 1/20 0.52
L3MBTL1 Q9Y468 1/20 0.46
NPSR1 Q6W5P4 2/20 0.45
GAA P10253 1/20 0.44
KMT2A Q03164 5/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
NPC1 O15118 1/20 0.44
STS P08842 1/20 0.43
CYP1A2 P05177 2/20 0.43
GLA P06280 1/20 0.43
TSHR P16473 1/20 0.43
SIRT5 Q9NXA8 1/20 0.42
LMNA P02545 2/20 0.42
POLB P06746 1/20 0.42
ELANE P08246 1/20 0.41
MAOB P27338 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4069238 0.87 MAPT (0.57) MAPTRAB9AHPGDL3MBTL1NPSR1
SCHEMBL17479477 0.80 GSK3B (0.56) KMT2ASMN1; SMN2
SCHEMBL22289601 0.80 ALDH1A1 (0.48) MAPTHPGDGAAKMT2ASMN1; SMN2
SCHEMBL28805020 0.75 MAPT (0.52) MAPTRAB9AHPGDL3MBTL1NPSR1
SCHEMBL28668806 0.75 MAPT (0.52) MAPTRAB9AHPGDL3MBTL1NPSR1
4-Nitrophenyl Methylcarbamate SCHEMBL31417181 0.75 MGLL (0.57) MAPTRAB9ANPSR1GAAKMT2A
SCHEMBL175551 0.74 MAPT (0.67) MAPTRAB9AHPGDL3MBTL1NPSR1
SCHEMBL10355780 0.74 MAPT (0.67) MAPTRAB9AHPGDL3MBTL1NPSR1
4-(Acetate)Acetophenone SCHEMBL1142839 0.74 MAPT (0.67) MAPTRAB9AHPGDL3MBTL1NPSR1
SCHEMBL12893245 0.74 ALDH1A1 (0.51) MAPTRAB9AHPGDGAAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3180317-A1 FACTOR XIa INHIBITORS Merck Sharp & Dohme Corp. (US) 2017-06-21 EP disclosed
WO-2016015593-A1 FACTOR XIa INHIBITORS MERCK SHARP & DOHME CORP. (US) 2016-02-04 WO disclosed