SCHEMBL17486102

SCHEMBL17486102

CC1(C)c2ccccc2-c2cc(-c3nc(-c4ccc(-c5cnc(-c6ccc7c(c6)C(C)(C)C(C)(C)C7(C)C)c(C#N)c5)cc4)nc(-c4ccc5c(c4)-c4ccccc4C5(C)C)n3)ccc21

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.33
NPSR1 Q6W5P4 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
KDM4E B2RXH2 3/20 0.32
HTT P42858 1/20 0.32
RXFP1 Q9HBX9 1/20 0.32
PDK2 Q15119 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
TNKS O95271 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
PIP4K2A P48426 1/20 0.31
LMNA P02545 1/20 0.30
THRB P10828 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17485971 0.83 HSD17B1 (0.34) ALDH1A1PDK2
SCHEMBL20805518 0.82 PIP4K2A (0.32) ALDH1A1NPSR1TDP1PIP4K2A
SCHEMBL17486186 0.78 CYP11B1 (0.31) ALDH1A1KDM4EHTTRXFP1LMNA
SCHEMBL19295172 0.78 ALOX5AP (0.39)
SCHEMBL19295140 0.76 PDK2 (0.34) PDK2
SCHEMBL17486246 0.76 HSD17B1 (0.33) ALDH1A1KDM4EPDK2L3MBTL1LMNA
SCHEMBL20805853 0.75 S1PR1 (0.34) NPSR1KDM4EPIP4K2ATHRB
SCHEMBL22986992 0.73 MEN1 (0.44) ALDH1A1NPSR1TDP1KDM4EHTT
SCHEMBL22037587 0.73 MEN1 (0.44) ALDH1A1NPSR1TDP1KDM4EHTT
SCHEMBL22914302 0.73 PDK2 (0.39) ALDH1A1PDK2CYP1A2CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3174890-B1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2019-03-13 EP disclosed
US-9853228-B2 Metal complexes MERCK PATENT GMBH (DE) 2017-12-26 US disclosed
US-20170250353-A1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2017-08-31 US disclosed
WO-2016015815-A1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2016-02-04 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170250353-A1 METAL COMPLEXES SOD1, AP1M1, AP3M1 ALDH1A1 3721/4885NPSR1 3952/4885TDP1 3464/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.