SCHEMBL17486117

SCHEMBL17486117

CC(C)c1ccc(-c2nc(-c3ccc(C(C)C)cc3)nc(-c3cnc(-c4ccc5c(c4)C4CCC5C4)c(C#N)c3)n2)cc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 2/20 0.36
CASR P41180 1/20 0.33
ERBB2 P04626 2/20 0.32
MAP3K12 Q12852 1/20 0.32
EGFR P00533 1/20 0.31
HPGD P15428 2/20 0.31
KDM4E B2RXH2 1/20 0.31
GPR119 Q8TDV5 1/20 0.31
S1PR1 P21453 7/20 0.31
XDH P47989 1/20 0.31
TLR9 Q9NR96 1/20 0.31
TLR8 Q9NR97 1/20 0.31
TLR7 Q9NYK1 1/20 0.31
KCNH2 Q12809 1/20 0.31
NPC1 O15118 1/20 0.30
ALDH1A1 P00352 1/20 0.30
POLB P06746 1/20 0.30
RAB9A P51151 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
S1PR2 O95136 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19295168 0.85 PPARA (0.33) KDM1ASMN1; SMN2
SCHEMBL20805777 0.81 CASR (0.33) KDM1ACASRKDM4ES1PR1TLR9
SCHEMBL17486287 0.76 CHRNA1 (0.34) KDM1AKDM4EALDH1A1
SCHEMBL19295180 0.76 IKBKB (0.35) KDM1ACASR
SCHEMBL20805776 0.76 CNR2 (0.32) KDM1A
SCHEMBL17486201 0.71 PDGFRB (0.32)
SCHEMBL17486052 0.69 DHODH (0.35)
SCHEMBL20805515 0.68 CYP11B1 (0.35)
SCHEMBL17486185 0.67 CYP11B1 (0.35)
SCHEMBL17485992 0.66 MEN1 (0.40) KDM1AHPGDKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3174890-B1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2019-03-13 EP disclosed
WO-2016015815-A1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2016-02-04 WO disclosed