SCHEMBL17486287

SCHEMBL17486287

N#Cc1cc(Br)cnc1-c1ccc2c(c1)C1CCC2C1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNA1 P02708 1/20 0.34
CHRNG P07510 1/20 0.34
CHRNB1 P11230 1/20 0.34
CHRNB2 P17787 1/20 0.34
CHRNB4 P30926 1/20 0.34
CHRNA3 P32297 1/20 0.34
CHRNA4 P43681 1/20 0.34
CHRND Q07001 1/20 0.34
CYP11B1 P15538 1/20 0.34
CYP11B2 P19099 1/20 0.34
JAK1 P23458 2/20 0.33
JAK3 P52333 2/20 0.33
MAPT P10636 2/20 0.33
TP53 P04637 1/20 0.33
JAK2 O60674 1/20 0.33
TYK2 P29597 1/20 0.33
KDM1A O60341 2/20 0.31
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
EP300 Q09472 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17486228 0.80 ALDH1A1 (0.34) CHRNB2CHRNA4JAK3MAPTALDH1A1
SCHEMBL17486224 0.80 KDM1A (0.35) CHRNB2CHRNB4CHRNA3CHRNA4MAPT
SCHEMBL17486117 0.76 KDM1A (0.36) KDM1AKDM4EALDH1A1
SCHEMBL17486201 0.76 PDGFRB (0.32)
SCHEMBL19295072 0.72 HSD17B1 (0.34) KDM1A
SCHEMBL17486043 0.71 CAMKK2 (0.36) JAK1JAK3JAK2TYK2
SCHEMBL19295078 0.70 IKBKB (0.35)
SCHEMBL17486281 0.69 PGR (0.37) CYP11B1CYP11B2
SCHEMBL17486170 0.68 SIGMAR1 (0.39) CHRNB2CHRNB4CHRNA3CHRNA4CYP11B1
SCHEMBL17486286 0.68 CYP11B1 (0.35) CYP11B1CYP11B2MAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3174890-B1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2019-03-13 EP disclosed
US-9853228-B2 Metal complexes MERCK PATENT GMBH (DE) 2017-12-26 US disclosed
US-20170250353-A1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2017-08-31 US disclosed
WO-2016015815-A1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2016-02-04 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170250353-A1 METAL COMPLEXES SOD1, AP1M1, AP3M1 CHRNA1 2662/4885CHRNG 2000/4885CHRNB1 3021/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.