SCHEMBL17486306

SCHEMBL17486306

CC(=O)c1cc(-c2ccc(-c3nc(-c4ccc(C(C)(C)C)cc4)nc(-c4ccc(C(C)(C)C)cc4)n3)cc2)cnc1-c1ccc2c(c1)C(C)(C)C(C)(C)C2(C)C

nearest known ligand 0.34

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 4/20 0.34
EPHB4 P54760 1/20 0.34
TEK Q02763 1/20 0.34
RARA P10276 1/20 0.33
RARB P10826 1/20 0.33
RARG P13631 1/20 0.33
ADORA3 P0DMS8 1/20 0.33
IKBKB O14920 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
CA12 O43570 1/20 0.32
CA9 Q16790 1/20 0.32
AKR1C2 P52895 1/20 0.32
AKR1C1 Q04828 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17485978 0.81 NPC1 (0.39) EPHB4TEKRARARARBRARG
SCHEMBL17486245 0.80 NPC1 (0.40) TRPV1EPHB4TEKRARARARB
SCHEMBL17486305 0.78 MAP4K4 (0.33) RARARARBRARGADORA3NPC1
SCHEMBL17486054 0.77 NPC1 (0.37) RARARARBRARGNPC1RAB9A
SCHEMBL17486123 0.76 TP53 (0.36) TRPV1RARARARBRARGNPC1
SCHEMBL17486017 0.76 SMN1; SMN2 (0.33) RARARARBRARGNPC1RAB9A
SCHEMBL17486302 0.74 TDO2 (0.37) TRPV1RARARARBRARGNPC1
SCHEMBL17486155 0.73 KDM4E (0.40) NPC1RAB9A
SCHEMBL19295157 0.71 NPC1 (0.36) RARARARBRARGNPC1RAB9A
SCHEMBL20805442 0.71 MELK (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3174890-B1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2019-03-13 EP disclosed
US-9853228-B2 Metal complexes MERCK PATENT GMBH (DE) 2017-12-26 US disclosed
US-9853228-B2 Metal complexes MERCK PATENT GMBH (DE) 2017-12-26 US disclosed
US-20170250353-A1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2017-08-31 US disclosed
US-20170250353-A1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2017-08-31 US disclosed
WO-2016015815-A1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2016-02-04 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170250353-A1 METAL COMPLEXES SOD1, AP1M1, AP3M1 TRPV1 1394/4885EPHB4 2639/4885TEK 4774/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.