SCHEMBL17488071

SCHEMBL17488071

Nc1nc2ccc(Nc3cc[nH]n3)cc2n1CCOc1ccc(OC(F)(F)F)cc1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CXCL8 P10145 1/20 0.42
NOD1 Q9Y239 1/20 0.42
KMT2A Q03164 1/20 0.42
DHFR P00374 2/20 0.41
NTRK1 P04629 3/20 0.38
KCNH2 Q12809 1/20 0.36
SCN5A Q14524 1/20 0.36
SCN9A Q15858 1/20 0.36
MCHR1 Q99705 3/20 0.36
EIF2AK2 P19525 1/20 0.36
MCHR2 Q969V1 1/20 0.35
ABL1 P00519 4/20 0.35
BCR P11274 4/20 0.35
IDH1 O75874 1/20 0.35
BRAF P15056 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17488072 0.94 CXCL8 (0.43) CXCL8NOD1KMT2ADHFRNTRK1
SCHEMBL17488202 0.82 NOD1 (0.46) CXCL8NOD1KMT2ADHFRNTRK1
SCHEMBL17488070 0.80 NOD1 (0.52) CXCL8NOD1KMT2ANTRK1SCN5A
SCHEMBL17488080 0.78 IDH1 (0.40) NTRK1MCHR1MCHR2IDH1
SCHEMBL17488185 0.76 IDH1 (0.41) NTRK1SCN9AMCHR1MCHR2IDH1
SCHEMBL17488184 0.75 IDH1 (0.42) MCHR1MCHR2IDH1
SCHEMBL17488075 0.73 KMT2A (0.52) CXCL8NOD1KMT2ANTRK1IDH1
SCHEMBL17488177 0.72 ALOX5AP (0.38) NTRK1SCN9AMCHR1ABL1BCR
SCHEMBL17488288 0.68 NTRK1 (0.41) CXCL8NOD1KMT2ANTRK1IDH1
SCHEMBL17488178 0.68 NTRK1 (0.42) CXCL8NOD1KMT2ADHFRNTRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016016421-A1 2-AMINO-BENZIMIDAZOLE DERIVATIVES AND THEIR USE AS 5-LIPOXYGENASE AND/OR PROSTAGLANDIN E SYNTHASE INHIBITORS INSTITUT PASTEUR KOREA (KR) 2016-02-04 WO disclosed