SCHEMBL17502172

SCHEMBL17502172

COC(=O)c1ccc(Sc2ccc(C#N)nc2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 1/20 0.45
MAPT P10636 8/20 0.43
CA1 P00915 2/20 0.42
CA2 P00918 2/20 0.42
ALDH1A1 P00352 5/20 0.42
KMT2A Q03164 1/20 0.42
MAPK1 P28482 3/20 0.42
KDM4E B2RXH2 6/20 0.41
POLB P06746 1/20 0.41
RAB9A P51151 2/20 0.41
NPC1 O15118 1/20 0.41
NFKB1 P19838 1/20 0.41
NFKB2 Q00653 1/20 0.41
RELA Q04206 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
L3MBTL1 Q9Y468 3/20 0.40
TDP1 Q9NUW8 1/20 0.40
CA12 O43570 1/20 0.40
CA7 P43166 1/20 0.40
CA9 Q16790 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL880697 0.84 MAPK1 (0.59) PTPN1MAPTCA1CA2ALDH1A1
SCHEMBL17502180 0.82 SLC22A12 (0.43) ALDH1A1KDM4ESMN1; SMN2L3MBTL1KCNQ3
Hydrochloric Acid SCHEMBL853571 0.82 MAPK1 (0.57) PTPN1MAPTCA1CA2ALDH1A1
SCHEMBL1169047 0.81 PTPN1 (0.50) PTPN1MAPTCA1CA2ALDH1A1
SCHEMBL25212412 0.80 TDP1 (0.49) MAPTCA1CA2ALDH1A1KMT2A
SCHEMBL25267522 0.78 MAPK1 (0.45) MAPTCA1CA2ALDH1A1KMT2A
SCHEMBL25216802 0.78 NNMT (0.51) PTPN1MAPTCA1CA2ALDH1A1
SCHEMBL25213750 0.78 ALDH1A1 (0.51) MAPTCA1CA2ALDH1A1KMT2A
SCHEMBL6575703 0.78 CA1 (0.61) MAPTCA1CA2ALDH1A1KMT2A
SCHEMBL25216660 0.78 ALDH1A1 (0.50) MAPTCA1CA2ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016022626-A1 HETEROCYCLIC CGRP RECEPTOR ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2016-02-11 WO disclosed