SCHEMBL17524949

SCHEMBL17524949

Nc1cnc(N2CCC3(CC2)C(=O)Nc2ncccc23)nc1

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CALCA P06881 5/20 0.41
CALCRL Q16602 9/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
TSHR P16473 1/20 0.37
HTR7 P34969 1/20 0.36
PARP1 P09874 1/20 0.35
OTUD7B Q6GQQ9 1/20 0.35
TNKS O95271 1/20 0.34
TNKS2 Q9H2K2 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17506417 0.85 CALCA (0.40) CALCACALCRLCYP3A4CYP2D6TSHR
SCHEMBL17524923 0.84 CALCA (0.41) CALCACALCRLHTR7OTUD7B
SCHEMBL1700112 0.81 CALCA (0.49) CALCACALCRLOTUD7B
SCHEMBL13806581 0.80 CALCA (0.46) CALCACALCRLOTUD7B
SCHEMBL16235885 0.79 CALCA (0.46) CALCACALCRLOTUD7B
SCHEMBL12655392 0.79 CALCA (0.47) CALCACALCRLOTUD7B
SCHEMBL12400699 0.79 CALCA (0.45) CALCACALCRLOTUD7B
SCHEMBL17524997 0.78 EGLN1 (0.43) CALCACALCRLHTR7
SCHEMBL17524906 0.78 CALCA (0.40) CALCACALCRLHTR7
SCHEMBL17525019 0.78 MAPK1 (0.41) CALCACALCRLCYP3A4CYP2D6TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016022644-A1 HETEROCYCLIC CGRP RECEPTOR ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2016-02-11 WO disclosed