SCHEMBL17524906

SCHEMBL17524906

Cc1cnc(N2CCC3(CC2)C(=O)Nc2ncccc23)cn1

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CALCA P06881 4/20 0.40
SMO Q99835 1/20 0.36
CALCRL Q16602 6/20 0.36
PTPN11 Q06124 4/20 0.36
HTR7 P34969 1/20 0.35
EGLN1 Q9GZT9 1/20 0.35
KCNH2 Q12809 2/20 0.35
OPRM1 P35372 1/20 0.34
OPRL1 P41146 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17524992 0.87 CALCA (0.39) CALCAHTR7KCNH2
SCHEMBL17524934 0.87 CALCA (0.39) CALCACALCRLPTPN11
SCHEMBL17524997 0.86 EGLN1 (0.43) CALCACALCRLHTR7EGLN1KCNH2
SCHEMBL17506417 0.83 CALCA (0.40) CALCACALCRLHTR7KCNH2
SCHEMBL17524937 0.82 ME2 (0.40) CALCACALCRLKCNH2
SCHEMBL17525014 0.81 CALCA (0.38) CALCACALCRLKCNH2
SCHEMBL17525112 0.81 SCN9A (0.43) CALCASMOCALCRLPTPN11
SCHEMBL1700112 0.79 CALCA (0.49) CALCACALCRL
SCHEMBL17524949 0.78 CALCA (0.41) CALCACALCRLHTR7
SCHEMBL13806581 0.78 CALCA (0.46) CALCACALCRLOPRM1OPRL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016022644-A1 HETEROCYCLIC CGRP RECEPTOR ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2016-02-11 WO disclosed