SCHEMBL17525944

SCHEMBL17525944

C[C@@]12CCCC1C1CCc3cc(C#N)ccc3C1CC2

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SHBG P04278 4/20 0.70
STS P08842 6/20 0.60
AKR1C3 P42330 1/20 0.54
ABCB11 O95342 3/20 0.48
HSD17B1 P14061 4/20 0.48
ESR1 P03372 6/20 0.45
ESR2 Q92731 5/20 0.45
HSD17B10 Q99714 4/20 0.45
LMNA P02545 3/20 0.45
PGR P06401 3/20 0.45
CYP3A4 P08684 3/20 0.45
AR P10275 3/20 0.45
SLC6A4 P31645 3/20 0.45
HTR2B P41595 3/20 0.45
SLC6A3 Q01959 3/20 0.45
AKR1B10 O60218 2/20 0.45
CYP1A2 P05177 2/20 0.45
SERPINA6 P08185 2/20 0.45
MAPT P10636 2/20 0.45
AKR1B1 P15121 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7864592 0.83 SHBG (1.00) SHBGSTSABCB11HSD17B1ESR1
SCHEMBL29643366 0.83 SHBG (1.00) SHBGSTSABCB11HSD17B1ESR1
SCHEMBL712443 0.83 SHBG (1.00) SHBGSTSABCB11HSD17B1ESR1
SCHEMBL172746 0.83 SHBG (1.00) SHBGSTSABCB11HSD17B1ESR1
SCHEMBL6695130 0.81 SHBG (0.75) SHBGSTSABCB11HSD17B1ESR1
SCHEMBL14048691 0.81 SHBG (0.46) SHBGSTSAKR1C3ABCB11HSD17B1
SCHEMBL6842205 0.80 AKR1C3 (0.49) SHBGSTSAKR1C3ABCB11HSD17B1
SCHEMBL13951936 0.80 STS (0.71) SHBGSTSHSD17B1ESR1ESR2
SCHEMBL15973298 0.80 AKR1C3 (0.53) SHBGSTSAKR1C3ABCB11HSD17B1
SCHEMBL15973296 0.80 STS (0.71) SHBGSTSHSD17B1ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2147014-B1 17ALPHA-SUBSTITUTED STEROIDS AS SYSTEMIC ANTIANDROGENS AND SELECTIVE ANDROGEN RECEPTOR MODULATORS ENDORECH INC (CA) 2016-02-17 EP disclosed