SCHEMBL17526328

SCHEMBL17526328

CCOC1CCCCc2ccccc21

nearest known ligand 0.56

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 4/20 0.56
GPR84 Q9NQS5 2/20 0.47
FFAR1 O14842 1/20 0.44
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.40
XBP1 P17861 1/20 0.40
HTT P42858 1/20 0.40
AKR1C3 P42330 1/20 0.39
AKR1C1 Q04828 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20433788 0.95 IDO1 (0.62) IDO1GPR84FFAR1ALDH1A1XBP1
SCHEMBL29890737 0.95 IDO1 (0.62) IDO1GPR84FFAR1ALDH1A1XBP1
SCHEMBL10340150 0.95 IDO1 (0.62) IDO1GPR84FFAR1ALDH1A1XBP1
SCHEMBL14461584 0.88 IDO1 (0.59) IDO1GPR84FFAR1
SCHEMBL19529546 0.82 GPR84 (0.59) IDO1GPR84FFAR1ALDH1A1HTT
SCHEMBL20433856 0.82 GPR84 (0.59) IDO1GPR84FFAR1ALDH1A1HTT
Acetic Acid SCHEMBL27529459 0.80 FFAR1 (0.52) IDO1GPR84FFAR1KDM4EALDH1A1
SCHEMBL8082622 0.78 IDO1 (0.62) IDO1GPR84FFAR1ALDH1A1KMT2A
SCHEMBL7326172 0.78 IDO1 (0.62) IDO1GPR84FFAR1ALDH1A1XBP1
SCHEMBL6689946 0.78 IDO1 (0.67) IDO1GPR84FFAR1ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2220061-B1 SPIRO-CONDENSED 1, 3, 4-THIADIAZOLE DERIVATIVES FOR INHIBITING KSP KINESIN ACTIVITY MERCK SHARP & DOHME (US) 2016-02-17 EP disclosed